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Cordycepin

Tier C — Watch / trade

Cordycepin

Danisco
Originator
-
First approval
-
Expiry (public)
No sales data
Peak sales
Small molecule
Type

Targets:Updating

Indications (approved):淋巴细胞减少症, Solid tumour, Lymphocytic leukaemia, Leukaemia

Regional status

US
No progress
1997-12-01
EU
-
China
Phase II
2025-12-01
Japan
-

Synthetic routes & intermediates3 routes

Originator routes × 1Optimised (non-patent) × 2Process routes × 0

Routes are ordered originator first, then optimised / process (non-patent) routes; each lists steps, overall yield and the intermediate table (code / CAS / name) — ready for supplier sourcing and RFQ. Rendered by this site from structured data; no third-party route graphics used.

OriginatorRoute 3Steps 4 · Total yield 1.04 g
CORD-00158-61-7CORD-01378-39-7CORD-01442867-77-6CORD-01562805-48-5CORD-01671196-28-6API · Cordycepin
CodeCAS No.Intermediate
CORD-00158-61-7Available(2R,3R,4S,5R)-2-(6-amino-9H-purin-9-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol
CORD-01378-39-7Available1,1,1-triethoxyethane
CORD-01442867-77-6((3aR,4R,6R,6aR)-6-(6-amino-9H-purin-9-yl)-2-ethoxy-2-methyltetrahydrofuro[3,4-d][1,3]dioxol-4-yl)methanol
CORD-01562805-48-5((2R,3S,4S,5R)-4-acetoxy-5-(6-amino-9H-purin-9-yl)-3-bromotetrahydrofuran-2-yl)methyl acetate
CORD-01671196-28-6((2S,4R,5R)-4-acetoxy-5-(6-amino-9H-purin-9-yl)tetrahydrofuran-2-yl)methyl acetate
OptimisedRoute 1Steps 3 · Total yield 36 g
CORD-00158-61-7CORD-0021026637-58-0CORD-00337731-72-9CORD-00437731-73-0API · Cordycepin
CodeCAS No.Intermediate
CORD-00158-61-7Available(2R,3R,4S,5R)-2-(6-amino-9H-purin-9-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol
CORD-0021026637-58-01-bromo-3-methyl-1-oxobutan-2-yl acetate
CORD-00337731-72-9(2R,3S,4S,5R)-2-(6-amino-9H-purin-9-yl)-4-bromo-5-(((2,4,4-trimethyl-5-oxo-1,3-dioxolan-2-yl)oxy)methyl)tetrahydrofuran-3-yl acetate
CORD-00437731-73-0(2R,3S,4R,5R)-2-(6-amino-9H-purin-9-yl)-4-bromo-5-(hydroxymethyl)tetrahydrofuran-3-ol
OptimisedRoute 2Steps 7 · Total yield 17.9 mg
CORD-005107-18-6CORD-006162825-77-6CORD-007162872-61-9CORD-008144867-90-3CORD-009—CORD-010164034-80-4CORD-01118055-46-4CORD-012162825-78-7API · Cordycepin
CodeCAS No.Intermediate
CORD-005107-18-6prop-2-en-1-ol
CORD-006162825-77-6(S)-oxiran-2-ylmethyl pivalate
CORD-007162872-61-9(S)-2-hydroxypent-4-yn-1-yl pivalate
CORD-008144867-90-3(S)-(2,3-dihydrofuran-2-yl)methyl pivalate
CORD-009-((2S,4R,5R)-4,5-dihydroxytetrahydrofuran-2-yl)methyl pivalate
CORD-010164034-80-4(2S,3R,5S)-5-((pivaloyloxy)methyl)tetrahydrofuran-2,3-diyl diacetate
CORD-01118055-46-4N-(trimethylsilyl)-N-(7-(trimethylsilyl)-7H-purin-6-yl)benzamide
CORD-012162825-78-7((2S,4R,5R)-4-acetoxy-5-(6-benzamido-9H-purin-9-yl)tetrahydrofuran-2-yl)methyl pivalate

Frequently asked questions

What are the approved indications of Cordycepin?

Approved indications include: 淋巴细胞减少症, Solid tumour, Lymphocytic leukaemia, Leukaemia.

When does the Cordycepin patent expire?

No public expiry year is available for Cordycepin yet; this page updates once verified.

How many synthesis routes are recorded for Cordycepin?

3 synthesis routes are recorded; the shortest is 3 steps with 36 g total yield. Intermediates in each route carry codes and CAS numbers.

Where can I buy Cordycepin intermediates?

2 intermediate CAS of Cordycepin are available through the Unibest supply network — see the route tables on this page and request a quote per CAS.

How do I get a quote for Cordycepin intermediates?

Open the CAS profile of the target intermediate from this page, or submit an RFQ directly — the CAS enters the matching flow automatically and the supply network responds with quotes.

Source: cross-verified data (structured fields only) · 2026-10-22