Patent-Cliff Blockbusters & Intermediate Opportunities

2028–2033 patent cliff mapped from cross-verified data sources, with actionable intermediate CAS lists

Curated LOE shortlist (SOP-reviewed) →

Hand-curated from this panorama: runway ≥ 3 years, barrier-scored, every CAS verified.

2556
Drugs
19
Tier A — Act now
101
Tier B — Position early
2436
Tier C — Watch / trade
21143
Intermediates →
Download full list (Excel: drug tiers + intermediates)
LOE opportunity profile · 3-step picker →

Pick region → your role → molecules of interest, generate a “what to buy / who is buying / how to pitch” profile, and match it directly against tracked customers and leads in the platform opportunity pool.

Browse by expiry year

Drugs losing exclusivity each year, with intermediates ready to source.

Therapeutic areas

Patent-cliff drugs grouped by indication and molecule.

Data digest

Monthly data digests →

Pipeline-derived monthly figures — verifiable, no marketing copy.

Tier A — Act now (peak sales ≥ $3B, expiry 2028–2031)

DrugGeneric nameOriginatorFirst approvalExpiryPeak($B)StepsInterm.
ApixabanApixabanBristol Myers Squibb2011202822.4▲640
SemaglutideSemaglutideNovo Nordisk2017203118.4*-0
IbrutinibIbrutinibPharmacyclics Llc201320279.78▲8163
EnzalutamideEnzalutamideUniversity of California, Los Angeles (UCLA)201220278.62▲515
RivaroxabanRivaroxabanBayer200820267.89▲948
Osimertinib MesylateOsimertinib MesylateAstraZeneca201520317.25▲729
EmpagliflozinEmpagliflozinBoehringer Ingelheim International Gmbh201420285.97▲825
Ruxolitinib PhosphateRuxolitinib PhosphateIncyte Corp201120285.88▲524
AbemaciclibAbemaciclibEli Lilly and Company201720295.72▲915
Dapagliflozin Propanediol/Metformin HydrochlorideDapagliflozin Propanediol/Metformin HydrochlorideAstraZeneca201420305.6*516
PalbociclibPalbociclibPfizer Inc.201520275.44▲952
Ribociclib SuccinateRibociclib SuccinateNovartis201720294.78▲914
OlaparibOlaparibAstraZeneca201420284.73▲613
Cariprazine HydrochlorideCariprazine HydrochlorideGedeon Richter Plc.201520294.47▲521
ZanubrutinibZanubrutinibBeiGene, Ltd.201920313.93▲1012
ApalutamideApalutamideJohnson & Johnson Innovative Medicine201820303.57▲1120
AcalabrutinibAcalabrutinibAstraZeneca201720303.52▲817
Lenvatinib MesilateLenvatinib MesilateEisai Co., Ltd.201520283.34▲918
BrexpiprazoleBrexpiprazoleOtsuka Pharmaceutical Co., Ltd.201520293.15▲318

Intermediate breakdown (all drugs with retrieved synthetic routes, by intermediate count)

Key intermediate CAS numbers registered in originator and optimised synthetic routes (cross-verified) — ready for supplier sourcing and RFQ.

Paclitaxel/Encequidar mesylate
CodeCAS No.
PACL-00127548-93-2
PACL-00217341-93-4
PACL-003103150-33-0
PACL-004102-94-3
PACL-005-
PACL-006114915-13-8
PACL-007114915-15-0
PACL-00898-88-4
PACL-009114915-17-2
Paclitaxel33069-62-4
(III)101438-1-a140-10-3
(IV)101438-1-a-
(VI)101438-1-a-
(VII)101438-1-a-
(VIII)101438-1-a-
(I)101438-2-a783-08-4
(II)101438-2-a13831-31-7
(III)101438-2-a146924-90-5
(IV)101438-2-a144790-01-2
(VI)101438-2-a132127-34-5
(VII)101438-2-a109-92-2
(VIII)101438-2-a201856-48-6
(X)101438-2-a201856-53-3
(XI)101438-2-a216094-54-1
View all 815 intermediates →
Paclitaxel6 steps
Paclitaxel
CodeCAS No.
PACL-00127548-93-2
PACL-00217341-93-4
PACL-003103150-33-0
PACL-004102-94-3
PACL-005-
PACL-006114915-13-8
PACL-007114915-15-0
PACL-00898-88-4
PACL-009114915-17-2
Paclitaxel33069-62-4
(III)101438-1-a140-10-3
(IV)101438-1-a-
(VI)101438-1-a-
(VII)101438-1-a-
(VIII)101438-1-a-
(I)101438-2-a783-08-4
(II)101438-2-a13831-31-7
(III)101438-2-a146924-90-5
(IV)101438-2-a144790-01-2
(VI)101438-2-a132127-34-5
(VII)101438-2-a109-92-2
(VIII)101438-2-a201856-48-6
(X)101438-2-a201856-53-3
(XI)101438-2-a216094-54-1
View all 815 intermediates →
Atorvastatin/Hydrochlorothiazide/Aspirin/Enalapril
CodeCAS No.
Enalapril-00164920-29-2
Enalapril-00213485-59-1
Enalapril-00382717-96-2
Enalapril-004147-85-3
Enalapril-00575847-73-3
Enalapril-006110-17-8
Enalapril-00753279-92-8
Enalapril-008120999-41-9
Enalapril-009138566-24-2
Enalapril-010-
Enalapril-0111142-20-7
Enalapril-01290315-82-5
Enalapril-01388767-98-0
Enalapril-01429375-30-2
Enalapril-015108428-39-3
Enalapril-0162812-46-6
Enalapril-01727544-35-0
Enalapril-01880828-26-8
Enalapril-019103377-40-8
Enalapril-02016652-71-4
Enalapril-021120924-94-9
Enalapril-02288098-09-3
Enalapril-023103-63-9
Enalapril-0243277-89-2
View all 251 intermediates →
Finerenone7 steps
Finerenone
CodeCAS No.
FINE-001959934-76-0
FINE-00221962-45-8
FINE-00365193-87-5
FINE-0041050477-39-8
FINE-00595306-64-2
FINE-0061050477-43-4
FINE-0071050477-44-5
FINE-0081050477-45-6
FINE-0091050477-27-4
(I)90859-10-a18368-64-4
(II)90859-10-a20173-49-3
(III)90859-10-a60323-96-8
(IV)90859-10-a79055-62-2
(VI)90859-10-a1663-67-8
(VII)90859-10-a107-12-0
(VIII)90859-10-a95306-65-3
(IX)90859-10-a41935-71-1
(X)90859-10-a1260663-96-4
(I)638294-1-a5394-63-8
(II)638294-1-a109-78-4
(V)638294-1-a1870824-80-8
(VIIIa)638294-1-a122-51-0
(VIIIb)638294-1-a,(VIIIb)638294-1-e78-39-7
(XII)638294-1-a2084136-51-4
View all 221 intermediates →
Docetaxel (Beihai)
CodeCAS No.
(I)140605-1-a-
(II)140605-1-a-
(I)140605-2-a2935-35-5
(II)140605-2-a333-27-7
140605-2-a24424-99-5
(III)140605-2-a141190-94-5
(IV)140605-2-a163061-19-6
(V)140605-2-a79265-30-8
(VI)140605-2-a163010-75-1
(VII)140605-2-a77-76-9
(VIII)140605-2-a163010-80-8
(IX)140605-2-a163010-82-0
(X)140605-2-a143527-70-2
(Ia)140605-3-a-
(Ib)140605-3-a71610-00-9
(Ic)140605-3-a251957-25-2
(IIa)140605-3-a78432-77-6
(IIb)140605-3-a,(IIb)140605-3-b76429-85-1
(IIc)140605-3-a199657-62-0
(IIIa)140605-3-a155556-72-2
(IIIb)140605-3-a-
(IIIc)140605-3-a-
(IVa)140605-3-a-
(IVb)140605-3-a-
View all 189 intermediates →
Docetaxel polymeric micelle (Samyang Biopharmaceuticals)
CodeCAS No.
(I)140605-1-a-
(II)140605-1-a-
(I)140605-2-a2935-35-5
(II)140605-2-a333-27-7
140605-2-a24424-99-5
(III)140605-2-a141190-94-5
(IV)140605-2-a163061-19-6
(V)140605-2-a79265-30-8
(VI)140605-2-a163010-75-1
(VII)140605-2-a77-76-9
(VIII)140605-2-a163010-80-8
(IX)140605-2-a163010-82-0
(X)140605-2-a143527-70-2
(Ia)140605-3-a-
(Ib)140605-3-a71610-00-9
(Ic)140605-3-a251957-25-2
(IIa)140605-3-a78432-77-6
(IIb)140605-3-a,(IIb)140605-3-b76429-85-1
(IIc)140605-3-a199657-62-0
(IIIa)140605-3-a155556-72-2
(IIIb)140605-3-a-
(IIIc)140605-3-a-
(IVa)140605-3-a-
(IVb)140605-3-a-
View all 188 intermediates →
Sertraline Citrate
CodeCAS No.
Sertraline Hydrochloride-001147514-83-8
Sertraline Hydrochloride-002147462-26-8
Sertraline Hydrochloride-003147462-27-9
Sertraline Hydrochloride-004147462-28-0
Sertraline Hydrochloride-005-
Sertraline Hydrochloride-006147462-29-1
Sertraline Hydrochloride-007147462-30-4
Sertraline Hydrochloride-008754157-48-7
Sertraline Hydrochloride-0091027935-40-5
Sertraline Hydrochloride-010791033-90-4
Sertraline Hydrochloride-011-
Sertraline Hydrochloride-012-
Sertraline Hydrochloride-013-
Sertraline Hydrochloride-0141093645-86-3
Sertraline Hydrochloride-015-
Sertraline Hydrochloride-016-
Sertraline Hydrochloride-017618910-81-9
Sertraline Hydrochloride-018-
Sertraline Hydrochloride-019-
Sertraline Hydrochloride-020-
Sertraline Hydrochloride-021-
Sertraline Hydrochloride-022-
Sertraline Hydrochloride-023-
Sertraline Hydrochloride-024-
View all 183 intermediates →
Atorvastatin strontium
CodeCAS No.
Atorvastatin-001-
Atorvastatin-00288-95-9
Atorvastatin-003-
Atorvastatin-004108998-83-0
Atorvastatin-005540-88-5
Atorvastatin-006222406-66-8
Atorvastatin-007110862-46-9
Atorvastatin-008222406-69-1
Atorvastatin-009222406-71-5
Atorvastatin-010222406-73-7
Atorvastatin-011134395-00-9
Atorvastatin-012793652-69-4
Atorvastatin-013222406-80-6
Atorvastatin-014-
Atorvastatin-015-
Atorvastatin-016-
Atorvastatin-017-
Atorvastatin-0181353049-81-6
Atorvastatin-019-
Atorvastatin-020-
Atorvastatin-021-
Atorvastatin-022838906-36-8
Atorvastatin-023-
Atorvastatin-024838906-52-8
View all 174 intermediates →
Atosiban acetate
CodeCAS No.
Atosiban-00129022-11-5
Atosiban-002-
Atosiban-003-
Atosiban-004109425-55-0
Atosiban-005-
Atosiban-006-
Atosiban-00771989-31-6
Atosiban-008-
Atosiban-009103213-32-7
Atosiban-010132388-59-1
Atosiban-011-
Atosiban-01271989-35-0
Atosiban-013-
Atosiban-014-
Atosiban-01571989-23-6
Atosiban-016-
Atosiban-017162502-65-0
Atosiban-018-
Atosiban-019-
Atosiban-020-
Atosiban-02127144-18-9
Atosiban-022-
Atosiban-02390779-69-4
Atosiban-024-
View all 171 intermediates →
Ibrutinib8 steps
Ibrutinib
CodeCAS No.
IBRT-0012215-77-2
IBRT-002330792-68-2
IBRT-003330792-69-3
IBRT-004330792-70-6
IBRT-005330786-24-8
IBRT-006143900-44-1
IBRT-0071022150-11-3
IBRT-008814-68-6
IBRT-0092380-63-4
IBRT-010151266-23-8
IBRT-01151067-38-0
IBRT-0121623-95-6
IBRT-0131574506-73-2
IBRT-0141574506-72-1
(I)461018-2-a83255-86-1
(IV)461018-2-a-
(VI)461018-2-a354-32-5
(VII)461018-2-a1441076-08-9
(VIII)461018-2-a1441076-09-0
(X)461018-2-a1441076-10-3
(II)461018-3-a109-77-3
(VII)461018-3-a4637-24-5
(II)461018-4-a541-41-3
(III)461018-4-a1652601-99-4
View all 163 intermediates →
Enalapril Maleate/Folic Acid
CodeCAS No.
Enalapril-00164920-29-2
Enalapril-00213485-59-1
Enalapril-00382717-96-2
Enalapril-004147-85-3
Enalapril-00575847-73-3
Enalapril-006110-17-8
Enalapril-00753279-92-8
Enalapril-008120999-41-9
Enalapril-009138566-24-2
Enalapril-010-
Enalapril-0111142-20-7
Enalapril-01290315-82-5
Enalapril-01388767-98-0
Enalapril-01429375-30-2
Enalapril-015108428-39-3
Enalapril-0162812-46-6
Enalapril-01727544-35-0
Enalapril-01880828-26-8
Enalapril-019103377-40-8
Enalapril-02016652-71-4
Enalapril-021120924-94-9
Enalapril-02288098-09-3
Enalapril-023103-63-9
Enalapril-0243277-89-2
View all 162 intermediates →
Dutasteride/Tamsulosin Hydrochloride
CodeCAS No.
Tamsulosin Hydrochloride-001122-84-9
Tamsulosin Hydrochloride-0023886-69-9
Tamsulosin Hydrochloride-003-
Tamsulosin Hydrochloride-004121565-95-5
Tamsulosin Hydrochloride-005112101-75-4
Tamsulosin Hydrochloride-006116091-64-6
Tamsulosin Hydrochloride-007103181-55-1
Tamsulosin Hydrochloride-008106133-20-4
Tamsulosin Hydrochloride-0093259-03-8
Tamsulosin Hydrochloride-01094-71-3
Tamsulosin Hydrochloride-01196-49-1
Tamsulosin Hydrochloride-0123250-73-5
Tamsulosin Hydrochloride-01386225-70-9
Tamsulosin Hydrochloride-014434312-10-4
Tamsulosin Hydrochloride-015-
Tamsulosin Hydrochloride-016-
Tamsulosin Hydrochloride-017754930-54-6
Tamsulosin Hydrochloride-018760126-31-6
Tamsulosin Hydrochloride-019112101-81-2
Tamsulosin Hydrochloride-020100-52-7
Tamsulosin Hydrochloride-021123-11-5
Tamsulosin Hydrochloride-022123-08-0
Tamsulosin Hydrochloride-023459-57-4
Tamsulosin Hydrochloride-024-
View all 154 intermediates →
Tadalafil/Tamsulosin
CodeCAS No.
Tamsulosin Hydrochloride-001122-84-9
Tamsulosin Hydrochloride-0023886-69-9
Tamsulosin Hydrochloride-003-
Tamsulosin Hydrochloride-004121565-95-5
Tamsulosin Hydrochloride-005112101-75-4
Tamsulosin Hydrochloride-006116091-64-6
Tamsulosin Hydrochloride-007103181-55-1
Tamsulosin Hydrochloride-008106133-20-4
Tamsulosin Hydrochloride-0093259-03-8
Tamsulosin Hydrochloride-01094-71-3
Tamsulosin Hydrochloride-01196-49-1
Tamsulosin Hydrochloride-0123250-73-5
Tamsulosin Hydrochloride-01386225-70-9
Tamsulosin Hydrochloride-014434312-10-4
Tamsulosin Hydrochloride-015-
Tamsulosin Hydrochloride-016-
Tamsulosin Hydrochloride-017754930-54-6
Tamsulosin Hydrochloride-018760126-31-6
Tamsulosin Hydrochloride-019112101-81-2
Tamsulosin Hydrochloride-020100-52-7
Tamsulosin Hydrochloride-021123-11-5
Tamsulosin Hydrochloride-022123-08-0
Tamsulosin Hydrochloride-023459-57-4
Tamsulosin Hydrochloride-024-
View all 140 intermediates →
Solifenacin Succinate/Tamsulosin Hydrochloride
CodeCAS No.
Tamsulosin Hydrochloride-001122-84-9
Tamsulosin Hydrochloride-0023886-69-9
Tamsulosin Hydrochloride-003-
Tamsulosin Hydrochloride-004121565-95-5
Tamsulosin Hydrochloride-005112101-75-4
Tamsulosin Hydrochloride-006116091-64-6
Tamsulosin Hydrochloride-007103181-55-1
Tamsulosin Hydrochloride-008106133-20-4
Tamsulosin Hydrochloride-0093259-03-8
Tamsulosin Hydrochloride-01094-71-3
Tamsulosin Hydrochloride-01196-49-1
Tamsulosin Hydrochloride-0123250-73-5
Tamsulosin Hydrochloride-01386225-70-9
Tamsulosin Hydrochloride-014434312-10-4
Tamsulosin Hydrochloride-015-
Tamsulosin Hydrochloride-016-
Tamsulosin Hydrochloride-017754930-54-6
Tamsulosin Hydrochloride-018760126-31-6
Tamsulosin Hydrochloride-019112101-81-2
Tamsulosin Hydrochloride-020100-52-7
Tamsulosin Hydrochloride-021123-11-5
Tamsulosin Hydrochloride-022123-08-0
Tamsulosin Hydrochloride-023459-57-4
Tamsulosin Hydrochloride-024-
View all 140 intermediates →
Drospirenone11 steps
Drospirenone
CodeCAS No.
(I)169995-1-a67372-65-0
(II)169995-1-a82543-07-5
(III)169995-1-a82543-09-7
(IV)169995-1-a82544-13-6
(V)169995-1-a82543-13-3
(VI)169995-1-a82543-14-4
(VII)169995-1-a82543-15-5
(VIII)169995-1-a82543-16-6
(IX)169995-1-a107-19-7
(X)169995-1-a82543-17-7
(XI)169995-1-a82543-18-8
(XII)169995-1-a,(XII)169995-1-b197721-70-3
(XIII)169995-1-a36865-41-5
(XIV)169995-1-a2707483-81-4
(XV)169995-1-a-
(XVI)169995-1-b1258501-10-8
(XVII)169995-1-b1258501-18-6
(XVIII)169995-1-b82546-55-2
(XIII)169995-2-a36255-44-4
(XIV)169995-2-a67372-66-1
(XV)169995-2-a67372-67-2
(XVI)169995-2-a67372-68-3
(XVII)169995-2-a67372-69-4
(XVIII)169995-2-a1774-47-6
View all 136 intermediates →
Atorvastatin Calcium Hydrate/Ramipril
CodeCAS No.
ATOR-001712-52-7
ATOR-0025754-35-8
ATOR-003110862-42-5
ATOR-00479-30-1
ATOR-005110862-44-7
ATOR-0067342-2-1
ATOR-007110862-45-8
ATOR-008110862-46-9
ATOR-0091429437-86-4
ATOR-010134523-00-5
ATOR-011125995-03-1
ATOR-0123886-69-9
ATOR-013-
ATOR-015134523-01-6
ATOR-016-
ATOR-017519-87-9
ATOR-018156051-77-3
ATOR-019156051-78-4
ATOR-02077-76-9
ATOR-021156051-79-5
ATOR-022156051-80-8
ATOR-023125971-96-2
ATOR-024156051-81-9
ATOR-025156051-82-0
View all 135 intermediates →
Tamsulosin Hydrochloride
CodeCAS No.
Tamsulosin Hydrochloride-001122-84-9
Tamsulosin Hydrochloride-0023886-69-9
Tamsulosin Hydrochloride-003-
Tamsulosin Hydrochloride-004121565-95-5
Tamsulosin Hydrochloride-005112101-75-4
Tamsulosin Hydrochloride-006116091-64-6
Tamsulosin Hydrochloride-007103181-55-1
Tamsulosin Hydrochloride-008106133-20-4
Tamsulosin Hydrochloride-0093259-03-8
Tamsulosin Hydrochloride-01094-71-3
Tamsulosin Hydrochloride-01196-49-1
Tamsulosin Hydrochloride-0123250-73-5
Tamsulosin Hydrochloride-01386225-70-9
Tamsulosin Hydrochloride-014434312-10-4
Tamsulosin Hydrochloride-015-
Tamsulosin Hydrochloride-016-
Tamsulosin Hydrochloride-017754930-54-6
Tamsulosin Hydrochloride-018760126-31-6
Tamsulosin Hydrochloride-019112101-81-2
Tamsulosin Hydrochloride-020100-52-7
Tamsulosin Hydrochloride-021123-11-5
Tamsulosin Hydrochloride-022123-08-0
Tamsulosin Hydrochloride-023459-57-4
Tamsulosin Hydrochloride-024-
View all 123 intermediates →
Ceftazidime/Tazobactam Sodium
CodeCAS No.
Ceftazidime-001141-97-9
Ceftazidime-002109-95-5
Ceftazidime-0031516-08-1,64-17-5
Ceftazidime-0045408-04-8
Ceftazidime-00562-56-6
Ceftazidime-00660845-81-0
Ceftazidime-00766338-99-6
Ceftazidime-00823877-12-5
Ceftazidime-00968672-65-1
Ceftazidime-01068672-66-2
Ceftazidime-011957-68-6
Ceftazidime-012127664-87-3
Ceftazidime-01373443-60-4
Ceftazidime-014110-86-1
Ceftazidime-01531461-04-8
Ceftazidime-016106134-67-2
Ceftazidime-01798445-42-2
Ceftazidime-01896752-43-1
Ceftazidime-0191040394-00-0
Ceftazidime-02089604-92-2
Ceftazidime-021102772-66-7
Ceftazidime-02286299-46-9
Ceftazidime-023120-78-5
Ceftazidime-02486299-47-0
View all 121 intermediates →
Efavirenz/Lamivudine/Tenofovir Disoproxil Fumarate
CodeCAS No.
LAMI-0013376-59-8
LAMI-00264904-47-8
LAMI-00353608-94-9
LAMI-004138760-43-7
LAMI-00571-30-7
LAMI-006143957-12-4
LAMI-00798-91-9
LAMI-0082032-35-1
LAMI-009163348-46-7
LAMI-01030163-03-2
LAMI-011143957-11-3
LAMI-012143957-14-6
LAMI-01389-78-1
LAMI-0141152495-30-1
LAMI-01526315-61-7
LAMI-01640018-26-6
LAMI-017-
LAMI-018147126-65-6
LAMI-019147027-10-9
LAMI-02068-11-1
LAMI-021298-12-4
LAMI-022138760-34-6
LAMI-023-
LAMI-024200396-19-6
View all 117 intermediates →
Rivastigmine Tartrate
CodeCAS No.
RIVAT-001105601-04-5
RIVAT-00288-10-8
RIVAT-003105601-20-5
RIVAT-0041243322-19-1
RIVAT-005139306-10-8
RIVAT-00742252-34-6
RIVAT-00832315-10-9
RIVAT-009121-71-1
RIVAT-010-
RIVAT-0111233378-72-7
RIVAT-0121233378-78-3
RIVAT-014855300-09-3
RIVAT-0151257519-35-9
RIVAT-016-
RIVAT-01710401-11-3
RIVAT-0181643442-41-4
(II)145089-1-a63720-38-7
(VI)145089-1-a-
(VII)145089-1-a530-62-1
(VIII)145089-1-a624-78-2
(IX)145089-1-a123441-03-2
(II)145089-2-a,(II)145089-2-e586-37-8
(III)145089-2-a122806-25-1
(IV)145089-2-a62409-13-6
View all 104 intermediates →
Emtricitabine/Rilpivirine Hydrochloride/Tenofovir Disoproxil Fumarate
CodeCAS No.
Tenofovir disoproxil phosphate-00178-95-5
Tenofovir disoproxil phosphate-00219141-39-0
Tenofovir disoproxil phosphate-00331618-90-3
Tenofovir disoproxil phosphate-0043167-63-3
Tenofovir disoproxil phosphate-005762-04-9
Tenofovir disoproxil phosphate-0063084-40-0
Tenofovir disoproxil phosphate-0071316848-77-7
Tenofovir disoproxil phosphate-00873-24-5
Tenofovir disoproxil phosphate-009180587-75-1
Tenofovir disoproxil phosphate-010206184-49-8,147127-19-3,147127-20-6
Tenofovir disoproxil phosphate-01135180-01-9
Tenofovir disoproxil phosphate-012201341-05-1
Tenofovir disoproxil phosphate-01315448-47-2
Tenofovir disoproxil phosphate-01414047-28-0
Tenofovir disoproxil phosphate-01516606-55-6
Tenofovir disoproxil phosphate-01660456-23-7,556-52-5
Tenofovir disoproxil phosphate-0174254-14-2
Tenofovir disoproxil phosphate-0184316-94-3
Tenofovir disoproxil phosphate-0191492978-64-9
Tenofovir disoproxil phosphate-0204316-93-2
Tenofovir disoproxil phosphate-0212799-16-8
Tenofovir disoproxil phosphate-022180587-74-0
Tenofovir disoproxil phosphate-02387-42-3
Tenofovir disoproxil phosphate-024598-31-2
View all 99 intermediates →
Tirzepatide18 steps
Tirzepatide
CodeCAS No.
Tirzepatide-00171989-33-8
Tirzepatide-002-
Tirzepatide-003-
Tirzepatide-004-
Tirzepatide-005-
Tirzepatide-006-
Tirzepatide-007-
Tirzepatide-008-
Tirzepatide-009-
Tirzepatide-010-
Tirzepatide-011-
Tirzepatide-012-
Tirzepatide-013-
Tirzepatide-014-
Tirzepatide-015-
Tirzepatide-016-
Tirzepatide-017-
Tirzepatide-018-
Tirzepatide-019-
Tirzepatide-020-
Tirzepatide-021-
Tirzepatide-022-
Tirzepatide-023-
Tirzepatide-024-
View all 96 intermediates →
Darunavir Ethanolate/Ritonavir
CodeCAS No.
RITO-0016372-14-1
RITO-00259830-60-3
RITO-003137649-69-5
RITO-00440635-67-4
RITO-005-
RITO-006177469-39-5
RITO-007144141-68-4
RITO-008144163-44-0
RITO-00998-80-6
RITO-010165315-39-9
RITO-011144163-97-3
RITO-012144164-11-4
RITO-013154212-61-0
RITO-014105-39-5
RITO-01533142-21-1
RITO-016115-08-2
RITO-01732955-22-9
RITO-01838585-74-9
RITO-0197693-46-1
RITO-020563-83-7
RITO-02113515-65-6
RITO-022534-07-6
RITO-0236306-52-1
RITO-024154212-60-9
View all 96 intermediates →
Ixabepilone15 steps
Ixabepilone
CodeCAS No.
IXAB-001192060-67-6
IXAB-0021119-51-3
IXAB-003219990-11-1
IXAB-004-
IXAB-005184917-63-3
IXAB-006219990-10-0
IXAB-007187283-47-2
IXAB-008-
IXAB-009-
IXAB-010-
IXAB-011302897-16-1
IXAB-012110-91-8
IXAB-01378-84-2
IXAB-0142403-55-6
IXAB-01579-03-8
IXAB-016106921-60-2
IXAB-017-
IXAB-01869739-34-0
IXAB-019187283-44-9
IXAB-020193146-29-1
IXAB-02193382-75-3
IXAB-02290600-20-7
IXAB-023208521-14-6
IXAB-024-
View all 96 intermediates →
View all 846 drugs with mapped synthetic routes →

Tier B — Position early

DrugGeneric nameOriginatorFirst approvalExpiryPeak($B)StepsInterm.
TirzepatideTirzepatideEli Lilly and Company2022203636.51▲1896
Nirmatrelvir/RitonavirNirmatrelvir/RitonavirPfizer Inc.2022-18.93▲-0
Bictegravir/Emtricitabine/Tenofovir Alafenamide FumarateBictegravir/Emtricitabine/Tenofovir Alafenamide FumarateGilead Inc2018-14.33▲740
Atorvastatin Calcium HydrateAtorvastatin Calcium HydratePfizer Inc.1996-13.69▲1158
LenalidomideLenalidomideCelgene Corporation2005-12.89▲522
BictegravirBictegravirGilead Inc-203312*47
Elexacaftor/ivacaftor/tezacaftorElexacaftor/ivacaftor/tezacaftorVertex Pharmaceuticals Incorporated2019-10.31▲-0
SofosbuvirSofosbuvirGilead Inc2013-10.28▲626
Dapagliflozin Propanediol MonohydrateDapagliflozin Propanediol MonohydrateBristol Myers Squibb2012-8.4▲516
UpadacitinibUpadacitinibAbbott Laboratories201920338.3▲34
Fluticasone Propionate/Salmeterol xinafoateFluticasone Propionate/Salmeterol xinafoateGSK1998-8.28▲-0
Rosuvastatin CalciumRosuvastatin CalciumShionogi & Co., Ltd.2002-7.05▲1055
Tafamidis MeglumineTafamidis MegluminePfizer Inc.2011-6.38▲527
ValsartanValsartanNovartis1996-6.05▲516
MontelukastMontelukastMerck & Co Inc1997-5.96▲1547
MolnupiravirMolnupiravir2021-5.68▲1085
PregabalinPregabalinPfizer Inc.2004-5.36▲832
Esomeprazole Magnesium HydrateEsomeprazole Magnesium HydrateAstraZeneca2000-4.43▲619
Pioglitazone HydrochloridePioglitazone HydrochlorideTakeda Pharmaceutical Company Limited1999-4.38▲528
Donepezil HydrochlorideDonepezil HydrochlorideEisai Co., Ltd.1996-4.35▲521
Candesartan CilexetilCandesartan CilexetilAstraZeneca1997-4.24▲956
Budesonide/Formoterol fumarate dihydrateBudesonide/Formoterol fumarate dihydrateAstraZeneca2000-3.8▲-0
Emtricitabine/Tenofovir Disoproxil FumarateEmtricitabine/Tenofovir Disoproxil FumarateGilead Sciences Inc2004-3.57▲-0
Sofosbuvir/VelpatasvirSofosbuvir/VelpatasvirGilead Inc2016-3.51▲626
Escitalopram OxalateEscitalopram Oxalate2002-3.49▲442
CelecoxibCelecoxibPfizer Inc.1998-3.33▲211
TelmisartanTelmisartanBoehringer Ingelheim International Gmbh1998-3.27▲835
TreprostinilTreprostinil2002-2.9▲1067
Nintedanib EsylateNintedanib EsylateBoehringer Ingelheim2014-2.83▲726
VenetoclaxVenetoclaxAbbVie201620302.79▲1131
Pemetrexed Disodium HydratePemetrexed Disodium HydrateEli Lilly and Company2004-2.79▲639
Emtricitabine/Tenofovir Alafenamide FumarateEmtricitabine/Tenofovir Alafenamide FumarateGilead Inc2016-2.76▲740
TadalafilTadalafilEli Lilly and Company2002-2.74▲517
DarolutamideDarolutamideOrion Corporation201920312.7▲69
Tofacitinib CitrateTofacitinib CitratePfizer Inc.201220282.46▲435
Simeprevir SodiumSimeprevir SodiumJohnson & Johnson Innovative Medicine2013-2.3▲624
ApremilastApremilastCelgene Corporation201420282.29▲525
IrbesartanIrbesartanSanofi1997-2.25▲629
Memantine HydrochlorideMemantine HydrochlorideMerz Pharma2002-2.25▲38
Dabrafenib MesylateDabrafenib MesylateGSK201320292.21▲612
MacitentanMacitentanActelion Pharmaceuticals Ltd2013-2.18▲1120
Dolutegravir SodiumDolutegravir SodiumGSK2013-2.18▲1741
Darunavir EthanolateDarunavir EthanolateTibotec2006-2.18▲1355
RisdiplamRisdiplamPtc Therapeutics Inc2020-2.13▲733
Lutetium (177Lu) vipivotide tetraxetanLutetium (177Lu) vipivotide tetraxetanRadiomedix Inc2022-1.99▲830
Cinacalcet HydrochlorideCinacalcet HydrochlorideAmgen2004-1.97▲526
Lurasidone HydrochlorideLurasidone HydrochlorideSumitomo Dainippon Pharma Co., Ltd.201020281.95▲423
LacosamideLacosamideUCB Pharma200820281.92▲335
Alectinib HydrochlorideAlectinib HydrochlorideChugai Pharmaceutical Co., Ltd.201420301.89▲1030
Ezetimibe/SimvastatinEzetimibe/SimvastatinMerck & Co Inc2004-1.88▲-0
Linagliptin/Metformin HydrochlorideLinagliptin/Metformin HydrochlorideBoehringer Ingelheim International Gmbh2012-1.86▲-0
Sugammadex SodiumSugammadex SodiumMerck & Co Inc200820281.84▲22
TolvaptanTolvaptanOtsuka Holdings Co Ltd200920281.84▲431
Edoxaban Tosilate HydrateEdoxaban Tosilate HydrateDaiichi Sankyo Co., Ltd.201120281.79▲1343
Dabigatran Etexilate MesylateDabigatran Etexilate MesylateBoehringer Ingelheim2008-1.75▲738
Bosentan HydrateBosentan HydrateF. Hoffmann-La Roche2001-1.71▲525
Esketamine HydrochlorideEsketamine HydrochloridePfizer Inc.199720291.7▲346
TelaprevirTelaprevirVertex Pharmaceuticals Incorporated2011-1.67▲655
Raltegravir PotassiumRaltegravir PotassiumMSD (Merck Sharp & Dohme)2007-1.67▲1113
Sodium Oxybate/Potassium Oxybate/Calcium Oxybate/Magnesium OxybateSodium Oxybate/Potassium Oxybate/Calcium Oxybate/Magnesium OxybateJazz Pharmaceuticals Plc2020-1.66▲-0
RiociguatRiociguatBayer2013-1.63▲913
EfavirenzEfavirenzBristol Myers Squibb1998-1.61▲632
Rabeprazole SodiumRabeprazole SodiumEisai Co., Ltd.1997-1.6▲49
TicagrelorTicagrelorAstraZeneca201020291.59▲955
CarfilzomibCarfilzomibOnyx Pharmaceuticals Inc201220291.57▲1031
Atazanavir SulfateAtazanavir SulfateBristol Myers Squibb2003-1.57▲836
MirabegronMirabegronAstellas Pharma Inc.201120291.54▲543
PaclitaxelPaclitaxelNational Institutes of Health (NIH)1992-1.54▲6815
Vortioxetine HydrobromideVortioxetine HydrobromideTakeda Pharmaceutical Company Limited2013-1.52▲519
Rilpivirine HydrochlorideRilpivirine HydrochlorideJanssen Therapeutics, Division of Janssen Products, LP2011-1.49▲428
Emtricitabine/Rilpivirine Hydrochloride/Tenofovir Disoproxil FumarateEmtricitabine/Rilpivirine Hydrochloride/Tenofovir Disoproxil FumarateGilead Sciences Inc2011-1.46▲799
Tezacaftor/IvacaftorTezacaftor/IvacaftorVertex Pharmaceuticals Incorporated2018-1.42▲-0
Sorafenib TosylateSorafenib TosylateOnyx Pharmaceuticals Inc2005-1.35▲514
DutasterideDutasterideGSK2001-1.35▲531
LinezolidLinezolidPfizer Inc.2000-1.35▲732
Solifenacin SuccinateSolifenacin SuccinateAstellas Pharma Inc.2004-1.34▲218
Levothyroxine SodiumLevothyroxine SodiumAbbVie2000-1.33▲420
Fluticasone PropionateFluticasone PropionateGSK1990-1.31▲528
VildagliptinVildagliptinNovartis2007-1.3▲625
Asciminib hydrochlorideAsciminib hydrochlorideNovartis2021-1.28▲48
Abacavir Sulfate/LamivudineAbacavir Sulfate/LamivudineViiv Healthcare2004-1.27▲-0
Saxagliptin HydrateSaxagliptin HydrateBristol Myers Squibb2009-1.25▲1150
Sunitinib MalateSunitinib MalatePfizer Inc.2006-1.24▲627
Budesonide/Formoterol fumarate/Glycopyrronium BromideBudesonide/Formoterol fumarate/Glycopyrronium BromideAstraZeneca2019-1.2▲555
Indacaterol Maleate/Glycopyrronium BromideIndacaterol Maleate/Glycopyrronium BromideNovartis2013-1.2▲421
Inclisiran sodiumInclisiran sodiumAlnylam Pharmaceuticals Inc2020-1.2▲-0
Canagliflozin/Metformin HydrochlorideCanagliflozin/Metformin HydrochlorideJohnson & Johnson Innovative Medicine201420291.11▲619
Varenicline TartrateVarenicline TartratePfizer Pharmaceuticals Ltd2006-1.11▲1019
DeferasiroxDeferasiroxNovartis2005-1.1▲28
Rivastigmine TartrateRivastigmine TartrateNovartis1998-1.09▲2104
Tenofovir Alafenamide FumarateTenofovir Alafenamide FumarateGilead Sciences Inc2016-1.07▲68
CannabidiolCannabidiolGw Pharmaceuticals Plc2018-1.06▲39
AxitinibAxitinibPfizer Inc.2012-1.04▲1131
AtogepantAtogepantMerck & Co Inc2021-1.04▲855
Sevelamer CarbonateSevelamer CarbonateGenzyme Corporation2000-1.04▲39
Cabozantinib S-malateCabozantinib S-malateExelixis Inc201220291.03▲721
FulvestrantFulvestrantAstraZeneca2002-1.03▲1234
LorlatinibLorlatinibPfizer Inc.201820301.02▲922
Olmesartan MedoxomilOlmesartan MedoxomilDaiichi Sankyo Co., Ltd.2002-1.02▲726
IvacaftorIvacaftorVertex Pharmaceuticals Incorporated2012-1.01▲832
Lopinavir/RitonavirLopinavir/RitonavirAbbVie2000-1.01▲-0

Tier C — Watch / fast-turnover trade

Vonoprazan Fumarate; Omeprazole; Finerenone; Brivaracetam; Pazopanib Hydrochloride; Azacitidine; Selpercatinib; Etelcalcetide Hydrochloride; Etonogestrel; Tamsulosin Hydrochloride; Ibandronate Sodium Hydrate; Voriconazole; Azilsartan; Bendamustine Hydrochloride; Ranolazine; Diroximel fumarate; Desvenlafaxine Succinate Hydrate; Posaconazole; Encorafenib; Bisoprolol Fumarate; Lumateperone tosylate; Sodium zirconium cyclosilicate; Linagliptin; Selumetinib sulfate; Cabazitaxel; Gefitinib; Nebivolol Hydrochloride; Avibactam Sodium/Ceftazidime; Dalfampridine; Icosapent ethyl; Liposomal bupivacaine; Regadenoson Hydrate; Ertapenem Sodium; Crizotinib; Risedronate Sodium Hydrate; Avatrombopag Maleate; Bimatoprost/Timolol Maleate; Lamivudine; Pimavanserin Tartrate; Alogliptin Benzoate; Brimonidine Tartrate/Timolol Maleate; Migalastat Hydrochloride; Ramipril; Avacincaptad pegol sodium; Omaveloxolone; Etoricoxib; Alpelisib; Eteplirsen; Entrectinib; Vonoprazan Acetate; Vibegron; Rotigotine; Lifitegrast; Tucatinib; Lubiprostone; Febuxostat; Exemestane; Zolmitriptan; Mirogabalin besilate; Fondaparinux Sodium; Ritonavir; Vemurafenib; Etravirine; Vildagliptin/Metformin Hydrochloride; Silodosin; Pimecrolimus; Avapritinib; Isavuconazonium Sulfate; Adefovir Dipivoxil; Fidaxomicin; Sumatriptan Succinate; Roxadustat; Voxelotor; Vismodegib; Givosiran; Tazobactam Sodium/Ceftolozane; Fezolinetant; Maribavir; Pralsetinib; Ripretinib; Selinexor; Remimazolam Besilate; Sotagliflozin; Relugolix; Erdafitinib; Alprazolam; Sevelamer Hydrochloride; Perampanel Hydrate; Orlistat; Mosapride Citrate; Ilaprazole; Ipragliflozin L-Proline; Latanoprost; Eptifibatide; Defibrotide sodium; Icotinib Hydrochloride; Indacaterol Maleate; Neratinib Maleate; Efinaconazole; Tedizolid Phosphate; Cobimetinib Fumarate; Binimetinib; Aclidinium Bromide; Diclofenac Sodium; Zuranolone; Azelastine Hydrochloride/Fluticasone Propionate; Lumasiran sodium; Ensifentrine; Trofinetide; Bepotastine besilate; Tegafur/Gimeracil/Oteracil Potassium; Naftopidil; Asenapine Maleate; Tafluprost; Lercanidipine Hydrochloride; Rucaparib Camsylate; Diquafosol Tetrasodium; Azelnidipine; Capmatinib Hydrochloride; Crisaborole; Olmesartan Medoxomil/Azelnidipine; Prucalopride Succinate; Glycopyrronium Bromide; Trospium Chloride/Xanomeline; Granisetron; Pacritinib Citrate; Memantine Hydrochloride/Donepezil Hydrochloride; Blonanserin; Fluticasone Propionate/Formoterol Fumarate Hydrate; Difamilast; Lanthanum carbonate hydrate; Oxcarbazepine; Trametinib; Fedratinib; Bilastine; Bupropion hydrobromide; Methylnaltrexone Bromide; Ixabepilone; Anagrelide Hydrochloride Hydrate; Omadacycline tosylate; Eravacycline; Aclidinium Bromide/Formoterol Fumarate Dihydrate; Canagliflozin Hemihydrate; Ciclesonide; Nitisinone; Ethinyl Estradiol/Norelgestromin; Pemigatinib; Evocalcet; Tofersen; Netarsudil Dimesylate; Romidepsin; Levosimendan; Daprodustat; Chidamide; Iguratimod; Formoterol Fumarate/Glycopyrrolate; Budesonide (Shire); Sivelestat Sodium Hydrate; Cefiderocol Sulfate Tosylate; Elobixibat Hydrate; Opicapone; Pralatrexate; Oxycodone Hydrochloride Hydrate; Mitiglinide; Landiolol Hydrochloride; Dordaviprone; Inotersen sodium; Fenofibrate; Fosnetupitant; Avanafil; Peramivir Hydrate; Dexamethasone Cipecilate; Emtricitabine; Timolol Maleate; Phenylephrine Hydrochloride; Valrubicin; Vadadustat; Lascufloxacin; Danoprevir Sodium; Fostamatinib disodium hexahydrate; Prasterone; Ephedrine Sulfate; Panobinostat Lactate; Amifampridine Phosphate; Miriplatin Hydrate; Elafibranor; Palovarotene; Glucosamine Hydrochloride; Entacapone; Remibrutinib; Delafloxacin; Safinamide Mesylate; Levomilnacipran Hydrochloride; Telavancin Hydrochloride; Ibuprofen; Folic Acid; Pilocarpine Hydrochloride; Gefapixant Citrate; Berotralstat; Sofpironium Bromide; Rilzabrutinib; Carotegrast methyl; Betrixaban; Lusutrombopag; Metformin Hydrochloride/Sitagliptin Hydrochloride; Flumatinib Mesylate; Riluzole (Aquestive Therapeutics); Cenobamate; Air polymer-type A; Amoxicillin/Omeprazole/Rifabutin; Asenapine transdermal therapeutic system(Hisamitsu Pharma); Lasmiditan hemisuccinate; Trifarotene; Ropinirole Hydrochloride transdermal (Hisamitsu Pharmaceutical); Tenapanor hydrochloride; Dolutegravir/Lamivudine/Tenofovir Alafenamide; Lefamulin; Pretomanid; Pexidartinib; Paclitaxel/Encequidar mesylate; L-Arginine hydrochloride/L-Lysine hydrochloride; Glucagon intranasal (Eli Lilly/Locemia Solutions); Cilastatin Sodium/Imipenem/Relebactam; Carrimycin; Bremelanotide; Quizartinib; Benvitimod; Drospirenone; PEG-Loxenatide; Tafamidis; Tecovirimat; Tegoprazan; Glycopyrrolate Tosylate; Dehydrated Alcohol Injection (Eton Pharmaceuticals); Moxidectin; Albuvirtide; Anlotinib Dihydrochloride; Atorvastatin Calcium Hydrate/Metformin Hydrochloride; Sitagliptin Phosphate Monohydrate/Ipragliflozin L-Proline; Lamivudine/Tenofovir Disoproxil Fumarate; Dexamethasone Implants(EyePoint Pharma); Efavirenz/Lamivudine/Tenofovir Disoproxil Fumarate; Atorvastatin/Hydrochlorothiazide/Aspirin/Enalapril; Fosravuconazole L-Lysine Ethanolate; Budesonide oral suspension (Dr Falk Pharma); Sodium ilaprazole; Angiotensin II; Macimorelin Acetate; Ertugliflozin; Sitagliptin/Ertugliflozin; Metformin Hydrochloride/Ertugliflozin; Dexpanthenol/Xylometazoline Hydrochloride; Noxiptiline hydrochloride; Ga-68 Edotreotide; Iron Isomaltoside; 6-[18F]Fluorodopa; Tadalafil/Tamsulosin; Polyethylene glycol/Sorbitol/Sodium Picosulfate; Hemoporfin; Carteolol Hydrochloride/Latanoprost; Telmisartan/Amlodipine Besylate/Hydrochlorothiazide; Grazoprevir Hydrate; Elbasvir; Paclitaxel Oral Solution (DAE HWA Pharmaceutical); Amlodipine Besylate/Fimasartan Potassium; Fimasartan potassium trihydrate/Rosuvastatin calcium; Dapagliflozin Propanediol Monohydrate/Saxagliptin Hydrochloride; Docetaxel polymeric micelle (Samyang Biopharmaceuticals); Oxymetazoline Hydrochloride/Tetracaine Hydrochloride; Gallium (68Ga) oxodotreotide; Betamethasone/Clotrimazole/Gentamicin Sulfate; Fluciclovine F 18; Olmutinib; Amlodipine Besylate/Tadalafil; Trelagliptin Succinate; Cangrelor Tetrasodium; Zabofloxacin Hydrochloride; Polmacoxib; Linagliptin/Empagliflozin; Atazanavir Sulfate/Cobicistat; Amlodipine Besylate/Perindopril Arginine; Dextromethorphan Hydrobromide/Chlorphenamine Maleate/Ammonium chloride; Paritaprevir/Ombitasvir/Ritonavir; Dasabuvir Sodium Hydrate; Ivabradine Hydrochloride/Metoprolol Tartrate; Rosuvastatin Calcium/Telmisartan; Darunavir Ethanolate/Ritonavir; Budesonide/Salmeterol xinafoate; Gemigliptin L-tartrate Sesquihydrate/Metformin Hydrochloride; Afamelanotide; Finafloxacin; Pasireotide Pamoate; Olmesartan Medoxomil/Amlodipine Maleate; Darunavir Ethanolate/Cobicistat; Olmesartan Medoxomil/Amlodipine orotate; Apatinib Mesylate; Methyl Salicylate/Levomenthol/Vitamin E/DL-Camphor; Sucroferric Oxyhydroxide; Lidocaine/Prilocaine cutaneous spray; Atorvastatin Calcium Hydrate/Irbesartan; Flutemetamol (18F); Allisartan Isoproxil; Olodaterol Hydrochloride; Solifenacin Succinate/Tamsulosin Hydrochloride; Conjugated Estrogens/Bazedoxifene Acetate; Diganan cross-linked sodium hyaluronate; Levamlodipine Besylate/Valsartan; Cetilistat; Cobicistat; Ibandronate Sodium Hydrate/Colecalciferol; Fenofibrate/Simvastatin; Rabeprazole Sodium/Metronidazole/Amoxicillin; Clarithromycin/Rabeprazole Sodium/Amoxicillin; Valsartan/Amlodipine Orotate; Afatinib Dimaleate; Lobeglitazone Sulfate; Valsartan/Lercanidipine Hydrochloride; Topiroxostat; Irbesartan/Trichlormethiazide; Bisoprolol Patches(Toa Eiyo); Fimasartan Potassium Trihydrate/Hydrochlorothiazide; Tilidine Hydrochloride; Pasireotide Diaspartate; Florbetapir(18F); Bixalomer; Metformin acetate; Radotinib Dihydrochloride; Artesunate/Pyronaridine Phosphate; Bupivacaine Hydrochloride/Fentanyl Citrate; Mifepristone/Misoprostol; Perchlozone; Diclofenac Sodium/Eperisone Hydrochloride; Arterolane maleate/Piperaquine Phosphate; Paroxetine/Alprazolam; Azilsartan Medoxomil Potassium/Chlorthalidone; Sibutramine maleate; Bisoprolol Fructoheptonate; Chung-Pa-Juhn; Alogliptin Benzoate/Pioglitazone Hydrochloride; Dutasteride/Tamsulosin Hydrochloride; Amlodipine Besylate/Bisoprolol Fumarate; Colecalciferol/Risedronate Sodium; Ibuprofen/Phenylephrine Hydrochloride; Tropisetron Citrate; Dienogest/Estradiol Valerate; Butylphthalide Injection(Cspc Ouyi Pharma); Amlodipine Besylate/Candesartan Cilexetil; Aliskiren; Ceftazidime/Tazobactam Sodium; Bepotastine Calcium Dihydrate; Metenkefalin/Tridecactide; Roxithromycin/Ambroxol Hydrochloride; Cinitapride Tartrate/Omeprazole; Miconazole/Metronidazole/Lidocaine; Clonidine Hydrochloride (Tris Pharma); Amlodipine Besylate/Telmisartan; Aztreonam lysine; Vinflunine Ditartrate; Hylastan; Fenofibric acid; Aspirin/Pseudoephedrine Hydrochloride; Rosilitazone Tartrate; Atorvastatin Calcium Hydrate/Ramipril; 18F-FP-CIT; Naproxen Sodium/Sumatriptan Succinate; Ticlopidine Hydrochloride/Ginkgo Biloba Leaf Dried Extract; Umirolimus; Sertraline Citrate; Prednisolone/Tetrahydrozoline Hydrochloride; Enalapril Maleate/Folic Acid; Ethambutol Hydrochloride/Rifampicin/Isoniazid; Menthol/Methyl Salicylate; Sitafloxacin Hydrate; Lodenafil carbonate; Clopidogrel Bisulfate/Aspirin; Atorvastatin strontium; Artesunate/Mefloquine Hydrochloride; Desvenlafaxine; Sodium Fluoride F-18; (R)-(+)-Rabeprazole sodium; Amlodipine Besylate/Olmesartan Medoxomil; Acetaminophen/Chlorphenamine Maleate/Methylephedrine Hydrochloride/Sulfogaiacol/Caffeine; Decitabine; Proxodolol hydrochloride/Pilocarpine Hydrochloride; Naltrexone controlled-release (Alkermes); Dextran/Calcium Chloride/Potassium Chloride/Sodium Chloride/Sodium lactate; Anidulafungin; Estradiol Valerate/Norethindrone Acetate; Cefoselis Sulfate; Betamethasone Dipropionate/Calcipotriol; S-pantoprazole sodium; Hydroxyethyl starch 130 / 0.4; Levamlodipine Besylate; Naloxone Hydrochloride/Oxycodone Hydrochloride Hydrate; Clevudine; Levocetirizine dihydrochloride/Pseudoephedrine Hydrochloride; Conivaptan Hydrochloride; Ibuprofen/Diphenhydramine Hydrochloride; Tolterodine Fumarate; Amodiaquine Hydrochloride; Nelarabine; Ivabradine Hydrochloride; Urinary Kallidinogenase; Inulin; Magnesium Isoglycyrrhizinate Hydrate; Naftifine hydrochloride/Ketoconazole; Amoxicillin Sodium; Tenofovir disoproxil phosphate; Formoterol Fumarate; Enalapril Maleate; Ceftazidime; Chlorphenamine Maleate; Tazobactam Sodium; Amlodipine Orotate; Lidocaine Hydrochloride; Metronidazole hydrochloride; Artesunate; Estradiol Valerate; Rifabutin; Imipenem; Xylometazoline Hydrochloride; Carteolol Hydrochloride; Fimasartan Potassium Trihydrate; Oxymetazoline Hydrochloride; Tetracaine Hydrochloride; Betamethasone; Clotrimazole; Metoprolol Succinate; Salmeterol xinafoate; Bazedoxifene Acetate; Simvastatin; Clarithromycin; Trichlormethiazide; Bupivacaine; Fentanyl; Mifepristone; Misoprostol; Eperisone Hydrochloride; Piperaquine Phosphate; Azilsartan Medoxomil Potassium; Chlorthalidone; Dienogest; Roxithromycin; Ambroxol Hydrochloride; Cinitapride Tartrate; Miconazole; Ticlopidine Hydrochloride; Ethambutol Hydrochloride; Rifampicin; Conteltinib; Betamethasone Dipropionate; Calcipotriol; Naloxone Hydrochloride; Ketoconazole; Docetaxel (Beihai); Pradefovir Mesylate; Inavolisib; Flurpiridaz F-18; Tasurgratinib; Levacetylleucine; Arimoclomol Citrate; Bortezomib Injection (Shilpa); Fulzerasib; Seladelpar lysine dihydrate; Vorasidenib; Gallium (68Ga) chloride/Germanium (68Ge) chloride; Benzgalantamine gluconate; Paliperidone Palmitate Injection(Ⅱ) (Luye Pharma); Deuterated ruxolitinib; Norethindrone Acetate/Ethinyl Estradiol; Chloral Hydrate Syrup(Hainan Pengkang Pharma); Cetirizine Hydrochloride Injection(Shandong Kexin Huiyi Pharma); Fultagliptin Benzoate; Epinephrine intranasal spray (ARS Pharmaceuticals); Bevifibatide Citrate; Naltrexone Hydrochloride Implants (Shenzhen Sciencare Medical Industries ); Thiotepa (Shorla Oncology); Rotigotine Microspheres for Injection(Luye Jiaao Pharma); Golidocitinib; Cofrogliptin; Rilertinib Mesylate; Envonalkib; Imetelstat; Lansoprazole and Sodium Bicarbonate Capsules(Xiamen Encheng Pharma); Sildenafil Citrate/Clomipramine Hydrochloride; Rezivertinib Mesylate; Allisartan Isoproxil/Amlodipine Besylate; Crisugabalin Besilate; Esomeprazole Magnesium and Sodium Bicarbonate Capsules(Xiamen Encheng Pharma); Mycophenolate mofetil oral (Azurity Pharmaceuticals); Upadacitinib Oral Solution(AbbVie); Lotilaner; Enavogliflozin/Metformin Hydrochloride; Dapagliflozin Propanediol Hydrate/Sitagliptin Phosphate Hydrate; Goserelin Microspheres for Injection(1-month long acting formulation,Luye Pharma); Pegmolesatide; Iruplinalkib; Retagliptin Phosphate; Anaprazole Sodium; Ritlecitinib tosylate; Nitroglycerin gel (Futura Medical); Vorolanib; Maritupirdine Hydrochloride; Sovateltide; Befotertinib Mesylate; Flotufolastat F-18; Durlobactam/Sulbactam sodium; Perfluorohexyloctane; Alfosbuvir; Triptorelin Acetate Microspheres for Injection(Shanghai Livzon Pharma); Sodium Oxybate Extended Release Oral Suspension (Avadel Pharmaceuticals); Risperidone long-acting injectable (Teva Branded Pharmaceutical); Niraparib Tosylate/Abiraterone Acetate; Potassium Sulfate/Anhydrous Sodium Sulfate/Anhydrous Magnesium Sulfate; Oxybutynin Hydrochloride (Hisamitsu); Leniolisib phosphate; Leritrelvir; Rezafungin acetate; Dexmedetomidine Hydrochloride Nasal Spray(Shanghai Hengrui Pharma); Zavegepant; Naloxone intranasal (Amphastar); Glumetinib; Glimepiride/Dapagliflozin Propanediol Monohydrate; Sparsentan; Keverprazan Hydrochloride; Bisoprolol Fumarate/Ramipril; Ganaxolone; Desidustat; Mitapivat sulfate; Orenetide; Tadalafil Oral Soluble Film(Qilu Pharma); Levornidazole Dispersible Tablets(Hunan Zhengtai Jinhu Pharma); Levornidazole Capsules(Hunan Zhengtai Jinhu Pharma); Rabeprazole Sodium/Sodium Bicarbonate; Clazosentan Sodium; Mitoxantrone hydrochloride liposome (CSPC ZhongQi); Daridorexant hydrochloride; Deuremidevir hydrobromide; Dalpiciclib Isethionate; Henagliflozin Proline; Levoketoconazole; Aildenafil Citrate; Fingolimod lauryl sulfate; Tadalafil/Finasteride; Pafolacianine Sodium; Olverembatinib; Nab-rapamycin; Sodium Phosphates Powder(Sichuan Jewelland Pharma); Paclitaxel Polymeric Micelles (Shanghai Yizhong Pharmaceutical); Triamcinolone Acetonide Suprachoroidal Injectable Suspension(Arctic Vision); Cefotaxime Sodium/Tazobactam Sodium; Chiglitazar Sodium; Varenicline Tartrate Nasal Spray(Oyster/Corxel ); Celecoxib/Tramadol Hydrochloride; Maralixibat Chloride; Vericiguat; Lazertinib Mesylate; Risperidone Microspheres for Injection (Ⅱ)(Luye Pharma); Surufatinib; Orelabrutinib; Emitasvir Phosphate; Sitagliptin Tartrate; Tirbanibulin; Ciprofol; Fluzoparib; TLX-591 companion diagnostic (Telix Pharmaceuticals); Setmelanotide Acetate; Olanzapine Oral Soluble Film(Jiangsu Hansoh); Lonafarnib; Ensartinib Hydrochloride; Sodium Sulfate/Magnesium Sulfate/Potassium Chloride; Losartan Potassium/Amlodipine Camsylate/Ezetimibe/Rosuvastatin Calcium; Amikacin liposomal (Insmed); Artemisinin (Oncotelic Therapeutics); Diperoxochloric acid; Hydrocortisone liquid (Eton Pharmaceuticals); Enarodustat; Bupivacaine/Meloxicam; Filgotinib Maleate; Glycopyrronium bromide/Neostigmine metilsulfate; Copper (64Cu) oxodotreotide; Clascoterone; Methocarbamol/Acetaminophen; Oliceridine fumarate; Bulevirtide Acetate; Edaravone/(+)-2-Decanol; Ravidasvir Hydrochloride; Lidocaine Cataplasms(Beijing Tide Pharma); Daclatasvir dihydrochloride/Asunaprevir/Beclabuvir hydrochloride; Tazarotene/Betamethasone Dipropionate; Piroxicam/β-Cyclodextrin; Repaglinide/Metformin Hydrochloride; Hydroxyethyl Starch 130/0.4 and Sodium Chloride; Aluminum Potassium Sulfate Hydrate/Tannic Acid; Boanmycin hydrochloride; Guaifenesin/Pseudoephedrine Hydrochloride; Omeprazole/Sodium Bicarbonate; Fluticasone propionate hydrofluoroalkane inhalation (GSK); Tribendimidine; Secretin; Gadoxetate Disodium; Ambroxol Hydrochloride/Clenbuterol Hydrochloride; Amlodipine Besylate/Atorvastatin Calcium Hydrate; Oxycodone; Calcium Citrate Malate; Clobetasol Propionate/Tretinoin; Reduced Glutathione Sodium; Macrogol 4000/Sodium Bicarbonate/Sodium Chloride/Potassium Chloride; Amlodipine Camsylate; Olanzapine/Fluoxetine hydrochloride; Belotecan Hydrochloride; Estradiol/Gestodene; Estradiol/Levonorgestrel; Amlodipine Maleate; Fosamprenavir Calcium; Fosfluconazole; Talaporfin Sodium; Etoprindole; Enalapril Maleate/Nitrendipine; Floxacillin sodium; Pazufloxacin Mesylate; Amrubicin Hydrochloride; Parecoxib Sodium; Fluocinolone Acetonide/Hydroquinone/Tretinoin; Atropine/Pralidoxime Chloride; Sulbactam sodium/Amoxicillin; Yttrium[90Y]; Dextrose/Sodium Chloride/Potassium Chloride/Sodium Bicarbonate; Trolamine; Chondroitin Sulfate Sodium/Allantoin/Vitamin E/Vitamin B6/Taurine; Coenzyme I; Neridronate Sodium; IG-RD-001; Eupatilin; Miltefosine; Cefonicid Sodium; Sultiame; Abacavir Sulfate/Lamivudine/Zidovudine; Carraghenates/Titanium dioxide/zinc oxide/Lidocaine; Arsenic Trioxide; Acitazanolast Hydrate; Candesartan Cilexetil/Hydrochlorothiazide; Glyburide/Metformin Hydrochloride; Cefazolin (B Braun Medical); Ioflupane (123I); Chlorhexidine gluconate/Isopropyl Alcohol; Maxacalcitol; Triptorelin Pamoate; Tolfenamic Acid; Cilastatin Sodium; Colesevelam Hydrochloride; Glycyrrhizin/Glycine/Cysteine Hydrochloride; Bulaquine; Alosetron Hydrochloride; Atosiban acetate; Cevimeline Hydrochloride Hydrate; Lafutidine; Technetium[99Tc] Methylenediphosphonate; Estradiol/Trimegestone; Dihydroetorphine Hydrochloride; Vincamine; Urapidil hydrochloride; Apomorphine Hydrochloride Injection (Britannia Pharmaceuticals); Bulaquine/Chloroquine Phosphate; Docosahexaenoic acid (DSM); Amoxicillin/Dicloxacillin sodium monohydrate; Auminium phosphate; Moherin; Benzbromarone; Arsenious Acid; Astaxanthin; Acetaminophen/Hydrocodone Bitartrate; Abacavir Sulfate; Tulobuterol; Leflunomide; Ganciclovir ophthalmic gel (Laboratoires Thea); Estradiol/Norethindrone Acetate; Ibuprofen/Levomenthol; Perindopril/Indapamide; Dermatan sulfate; Perflutren; Tirofiban Hydrochloride Hydrate; Bromfenac Sodium; Pramipexole Dihydrochloride Hydrate; Cefcamate Pivoxil Hydrochloride; Dydrogesterone/Estradiol; Ardeparin; Samarium (153Sm) lexidronam pentasodium; Nelfinavir Mesylate; Imiquimod; Naphazoline Hydrochloride/Chlorphenamine Maleate/Cyanocobalamin; Acetaminophen/Chlorphenamine Maleate/Dextromethorphan Hydrobromide/Pseudoephedrine Hydrochloride; Vidarabine Monophosphate; Lysine Tneophyllinate; Technetium [99mTc] Pentetate; Technetium [99mTc] L,L-Ethylenedicysteine; Indigo Carmine; Technetium[99mTc]Methylene diphosphonate; Technetium[99mTc]Succimer; Technetium [99mTc] Etifenin; Methylenediphosphonate/Stannous Chloride; indirubin; Technetium [99mTc] Phytate; Estradiol Valerate/Levonorgestrel; L-Phencynonate Hydrochloride; Lornoxicam; Acetylkitamycin; Luminol sodium; Tetrachlorodecaoxide; Kanglaite; Pilocarpine Hydrochloride (Allergan); Plazomicin sulfate; Pretomanid/Linezolid; RSC-1001; NVG-291; SBK-001; [225Ac]Ac-FL-261; RX-608; YMI-024; SMF-216; FXR-0906; Alpha-lactalbumin-oleic acid (Azanta); NBI-1117567; RXC-008; ONO-4578; Istaroxime; HKGM-453; PRO-1562; AD-233; TT-01488; FHD-286; VSA-012; Nilotinib Transdermal (KeifeRx); ALX-1; 64CU-DOTA-ECL1i; TQA-3605; H889A; VV-913; 64Cu-TR2205; HDNMGPTB-0226; [18F]FIDT-10b; JYP-0035; 68Ga-FAPI/18F-FDG; RO-7568282; HTX-201; AZD-6234; PL-3301; [18F]BF3-BPA; ND-003 (NewDEL Biotech); DDY-391; rupatifen fumarate (Fujian Mindong Rejuvenation Pharmaceutical/Fujian Institute of Microbiology); YKRH-00020; RFUS-188; KIT-2014; Secutrelvir; ABI-6250; APSTZD; Lumekefamide; GUB-014295; ARD-001; EA-230; Inobrodib; ZOC-2019619; VV-119; RG-6457; SYH-2085; OTR-8100; JKN-2501; SAL-0145; HSK-50042; XH-S003; CB-275; Domatinostat/Sirolimus; J-147; Zopocianine; TQD-3524; BH015; Colistimethate E2 sodium (Jiangsu Chia Tai-Tianqing Pharmaceutical); GDC-3280; HRS-9821; SRG-514; HSK-42360; PAX-1-001; Timolol Maleate Gel (Aucta Pharmaceuticals); ANS-02; nL-TARDB-002; Nivegacetor; RHNGLYOPH-0126; SHC-013; PRTX-007; Elismetrep; APG-157; HSK-31679; Rentosertib; BI-3034701; ZL-85-FA; [68Ga]BED003; S-233107; OD-001; LN-016; ENT-201; BRM-411; JMKX-000197; UBT-251; 68Ga-PSMA-0057; Selnoflast; GBI-268; RAP-219; DN-022150; Atebimetinib; MEX-CD1; BLU-924; NIO-752; TQC-3927; AZD-2287; Cleminorexton; Tacrolimus (VIVUS); HQ-2216; BSDO-2301; HDY-015; ERX-1000; TR-115; SIR9900; DAT-2645; YJ001; Privosegtor; PTH-IA; KET-AD; HL-300; MI-078; ABS-1230; DA-020; HRS-7058; naringin (Guangdong Zhongsheng Pharmaceutical/SCCIP/Sun Yat-Sen University); SCAI-005; CZ-012; SYH-2059; DX-243; Epinephrine inhalation aerosol (Kokua Pharma); LY-4395089; AZD-2265; BBI-001; HW-091077; LBS-007(Beijing Cro); Zn-Telomir; Proline-rich peptide hydrogel (Complutense University Of Madrid); SY-002 (Jiacheng Biomedical Technology); HS-10506; YKYY-029; BI 3000202; LN-003; Azenosertib; [11C]CS1P1; IMBZ1-8-g; MK-7762; Methylone; Abenacianine; TQ-B3234; Ropivacaine Extended-Release Microspheres (Yichang Humanwell); SC-0032; Pociredir; NS-035; UX-016; Rifabutin (BioVersys); HRS-6208; E2086; TAN-118; WD-890; QLS-111-FDC; Enicepatide; Tacrolimus (novaliq); GXV-813; HRS-1780; XTYW-007; TGM-312; ABSK-141; Gemcitabine Hydrochloride/Docetaxel; HB-5; ALN-2232; SNB-101; RBD-7022; TB511; BEBT-701; Butyrate Liquid; MLD-10; Terbium 161 DOTATATE PRRT; ATR-258; NTX-1024; CMS-D002; [18F]FPyQCP; ELV-001 (Elevara); Linepemat; SB-4826; Cemsidomide; Setidegrasib; NBI-1117570; LY-4065967; Apecotrep; TRG-200; HS-10542; Flonoltinib maleate; BL-0020; EXV-801; EXV-801/Dextromethorphan Hydrobromide; MOTS-c; LTI-03; Melanotan II; Bepecin; Nitrous oxide; MDR-001; Kamuvudine-9; Kamlanoflast; T-10430; EIK1005; SPN-821; INI-2004; HW-N2001; Nenocorilant; XNW-34017; Butylidenephthalide; JNJ-88545223; HRS-9563; DYTH-201; RAG-17; ZD-526; QLG-1194; Antisense Oligonucleotides (EveryONE Medicines); Psilocin Mucate; Amifostine for nasoduodenal delivery (Xerient Pharma); DNN.65.21.005; K110-42; Bupivacaine/Celecoxib; BAFA; Platelet membrane coated resiquimod nanoparticles (Cello Therapeutics); HRS-9057; Praziquantel / repurposed undisclosed anti-inflammatory drug (Drugs for Neglected Diseases initiative); BI-882370; Vopenfasinib; ACCG-2671; HBW-004285; 177Lu-PSMA-0057; TYK-01054; KN-510; KN-713; Budesonide Delayed-Release Tablets(Triastek); DNV-001; ECC-0509; ECC-4703; Viroxavir marboxil; MY-009; Vepugratinib; TM-471-1; 4-methylumbelliferyl trimebutine sulfate; VMD-3866; Atumelnant; S-337395; 18F-LNC1007; FT-2109; Minoxidil (Eurofarma Laboratorios); NLS-133; PH-15; Linafexor; Cordycepin; RJ-4287; BB-102; KH-001 (Kanna Health); Oxipurinol (XORTX Therapeutics); Florbetaben; Amezalpat; CL-197; LY-3537021; Oxandrolone subdermal (Stin Pharma); GEN-725; ICP-322; CRN-09682; Debio-4126; HE-009; HRS-1301; SAL-0140; LL-10; ABP-1011-T; KT-621; Asuptegravir; SL-1002; JKN-2301; JKN-2403; nL-ATN1-001; LAD-191; Anti-GD2-800CW; Trans-resveratrol (Jupiter Orphan Therapeutics); SV-001; RN-3161; SION‑719; HRS-7450; VES-001; RTN-001; SS-001(Suzhou Pairui Biotech); HRS-5632; UA-021; NS-136; 99mTc-ZHER2:41071; GSK-5460025; HRS-7085; ALDP-001; ABP-007; Macupatide; BM-2216; Quabodepistat; Brenipatide; S1B-509; BPC-2001; Bimatoprost-Drug Ring System (Spyglass Pharma); PTP-01; LY-3938577; AM-1002; H01; Buccal Dexmedetomidine (Reconnect Labs); OC-1; LDR-2402; bis-octanoyl (R)-1,3-butanediol (C8 ketone di-ester); Fudotinib; NEMO-103; TER-2013; GFH-276; AQW-051; RK-4; H-018; XJN-010; Muvalaplin; Methylphenidate (Inspirion); TQC-3721; HSK-47388; TQB-3201; ODS-101; TDM-Atop-01; Pracytarabine; T-1101; ENTR-601-45; Zilebesiran; Deudextromethorphan/Bupropion Hydrochloride; Dexmedetomidine hydrochloride microneedle patch(Guangzhou Novaken Pharma); Onvuzosiran; nL-PRPH2-001; TQB-3455; KYN-5356; CP-383; KYAH02-2016-078; 177Lu-NI-FAPI; Sacubitril/Valsartan Sodium Hydrate/Amlodipine; Elsunersen; AHB-137; HRS-7249; Hydrochloroquine; Deziglipel; Pt(0506)101; Repinatrabit; L-Adrenaline Brtartrate; BHB-1893; CTO-0308; PBK_M2502; LZHG-2403; Neracorvir; HRS-8080; Surzetoclax; SG-1; JKN-2304; Valganciclovir; NS-041; Paclitaxel Polymeric Micelles(Tumor Research Institute Chinese Academy Of Medical Sciences); Purinostat Mesylate; SC-101; Pidnarulex; TCIC-001; DZD-6008; Sutetinib Maleate; Pevifoscorvir Sodium; Cilostazol/Borneol; [F-18]Flornaptitril; S1B-408; HRS-1738; TAVT-119; TAVT-45; MT-501; GW-5282; Spermidine; ALKN-001; VK-2735; APL-3007; Prospidium chloride(Research Institute for Physical Chemical Problems of the Belarusian State University); H-021; OAB-14; PF-07328948; RAY-1225; LN-020; PS-101; Bleximenib; Zorevunersen; LT-002-158; ORC-13661; OD-07656; Paclitaxel cationic liposomes for injection(CSPC Zhongqi Pharma); SYHX-1901; VP-001; QR-059; SY-5933; Oxytocin/Estrogen; ABP-745; QLC-1101; DT-216; Bucillamine ((Intravenous); Capsaicin (Centrexion Therapeutics); STC-004; SKY-0515; R-Ketamine Hydrochloride Nasal Spray(Sichuan Purity Pharma); PRT-042; FXS-4640; T-168; BDB-001 (Eikon Therapeutics); EMP-01; Direclidine; INM-176; HS-10501; EXT-608; STC-15; Trichostatin A; Meglumine Sodium Succinate; DMX-101 (DIMERx); ONO-2020; HRS-6768; HRS-6719; INR-102; ALC-2203; HY-0902; 225Ac-LNC1011; Ezetimibe/Rosuvastatin Calcium/Candesartan Cilexetil/Amlodipine; Candesartan Cilexetil/Rosuvastatin Calcium/Ezetimibe; Dextromethorphan/Lidocaine; BG-136; Tacabrutideg; Omilancor; TRD-205; Suramin sodium (Kuzani Pharmaceuticals); ASI-02; Bemnifosbuvir/Ruzasvir; LND-101; LV-232; ECI-830; SASS-001; LNK-01002; INM-755; Kesonotide; Camprenstat; Brexanolone (Lipocine); QCZ-484; Zabalafin hydrogel (Alphyn Biologics); SRSD-216; ZG-001(Zhigen); ALD-102; TNG456; LLX-424; AUR-103; PF-08653945; Technetium [99mTc]-H7ND; R-Ketamine Hydrochloride Nasal Spray(Jiangsu Nhwa Pharma); ALN-4324; Tacrolimus (MedinCell); NTRX-07; Simmitinib; Padoprazan; CIL-001; GLK-401; OMS-405; BW-20805; Roginolisib; Semaglutide(Zhejiang Apeloa Kangyu Pharma); Oruvestat; 177Lu-LNC1011; NTX-001; HLX-1502; Salbutamol metered-dose inhalation(AstraZeneca); Pocenbrodib; [203-Pb] VMT-NET; HRS-8179; Ozone; Ulacamten; HLD-0915; Gabapentin/nabilone (PleoPharma); Levofloxacin/ketorolac trometamol (NTC); NTC-011; NTC-041; RSS-0343; ABP-1019-A; CGT-4859; Osavampator; Intravenous Melatonin (Cessatech); Carvedilol sulfate; H001; DWC-202314; TAR-0520; DWC-202404; RBS-2418; NEU-411; ONO-1110; SQ-727; Cirtuvivint; AERO-001; AERO-002; Glycopyrrolate/indacaterol (AeroRX Therapeutics/HCmed); Afamelanotide (Alys Pharmaceuticals); LPM-3770164; EOM147; NTP-42; I-025-A; HRS-2189; SRD-4610; B-007A; Cevimeline Ophthalmic Solution (BioTheraVision); CR999C1701L1; CR999K1601L1; Deuterated psilocybin analog; Enrupatinib; AMOR-1; GSK-4418959; Quemliclustat; HG-146; Sapanisertib/Serabelisib; Fosmanogepix; Lysergic acid diethylamide (Mind Medicine/The University Hospital of Basel); JMKX-003002; 177Lu-D7ND; RBD-1006; Cilnidipin (Aisa Pharma); GCWB-204; GCWB-211; GCWB-212; GCWB-213; IkT-001Pro; TAX-2; BP-102; Fexlamose; Daniluromer; 18F-FAPI; Soficitinib; SCR-6852; NTCB01-1; Grammidin; Lavengratinib; Lumipodlin; Naperiglipron; FC-084-CSA; QB0208-1; Carbon Nanoparticle-Loaded Iron; IG-3018; EV-25; Cetirizine Amidine Sodium; Betamethasone/Desloratadine (Laboratorios Silanes); RNK-08954; FLD-103; VB-15010; lartesertib; SIPI-2011; STC-007; SAL-0120; Simepdekinra; NX210c; PEG-Irinotecan; RS-113; Ponometrep; Lenacapavir/Islatravir; ACR-2316; Phosphocreatine; APG-2449; Emrusolmin; JIN-A04; Soquelitinib; RBM 39 targeting therapeutic (Recursion Pharmaceuticals); TRQ-001 Triquetra Medicines AB; Cariprazine hydrochloride (Chengdu Kanghong Pharmaceutical); Honokiol liposome lyophilized powder for injection (Jinrui Foundation); ZSP-0678; AIP-303; Florensocatib; STX-241; Buprenorphine depot (Alar Pharmaceuticals); SR-750; Hosu-53; DA-001 (Applied Biology); LP-118; Simmitinib hydrochloride; MAX-10181; Controlled-Ileocolonic-Release Nicotinamide (CICR-NAM); AG-1705; CM-9241GRU; PH-797904; MR-145-02; AG1901; Ubiquinol (Nobelpharma); MPB-1523; IGS-A0302; Weersuntinib; SN 38 loaded biodegradable nanofiber (Cebiotex); Lenacapavir pacfosacil; Lepetegravir; Lepetegravir/lenacapavir pacfosaci; Fluocinolone acetonide (FA) extended release(Eclipse Life Sciences); Modzatinib; 18F-Fluoromisonidazole; CT-7439; XS-02; RVP-001; ITU-512; EVO-756; SMP-3124LP; Synthetic psilocybin(Ceruvia Lifesciences); CG-0255 (PO); EPI-SK17; STAT-201; CYTO-200 AIMS™ Program; 18F-LNC1016; Visepegenatide; Deoxythymidine/Deoxycytidine; Olgotrelvir; Henagliflozin/metformin/retagliptin (Shandong Shengdi); Mifanertinib Maleate; Nerandomilast; Timolol maleate gel (Merson Pharma); Mufemilast; Imlunestrant Tosylate; Paltusotine; Lidocaine patch transdermal (D. Western Therapeutics Institute/MEDRx); Elamipretide; Bumetanide nasal spray (Corstasis Therapeutics); Gemcitabine controlled release (TARIS Biomedical); Zeprumetostat; Sepetaprost; Vornorexant; Donidalorsen; Dirozalkib; Cyclobenzaprine HCl sublingual tablets (Tonix Pharmaceuticals); Nor Ursodeoxycholic Acid; Brensocatib; Zongertinib; Aceclidine hydrochloride; Tegomil fumarate; Amlodipine Oral Solution (Brillian Pharma); Risperidone oral soluble Pellicles(Qilu Pharma); Tunodafil Hydrochloride; Sebaloxavir Marboxil; Elinzanetant; Lisaftoclax; Sebetralstat; Ifupinostat Hydrochloride; Amisulpride Orally Disintegrating Tablets(Shanghai Zezheng Bio-pharma); Tizanidine Hydrochloride(Sichuan Credit Pharma); Tibremciclib Tartrate; Octreotide chloride; Nilotinib Tartrate; Garsorasib; Sulopenem etzadroxil/Probenecid; Momelotinib Dihydrochloride; Irinotecan liposomal (CSPC); Motixafortide; Sunvozertinib; Tolvaptan Sodium Phosphate; Voclosporin; Molidustat Sodium; Anamorelin Hydrochloride; Olanzapine Oral Soluble Film(Qilu Pharma); SGN-101; Egalognastat; HJ-787; WVE-006; SPH-5030; BMS-986470; RTP-026; Sitafloxacin Fumarate; SJP-0170; Radiation injuries protective agent(RadioMedix); BR1019; Nanocurcumin (Tehran University of Medical Sciences); YR-001; SRP-1001; Golcadomide; Quinolisin; QLG-2198; 166-Ho microspheres; DT-678; 68Ga-NY104; 3HP-2827; Vicadrostat; Isoprocin glutarate; Cadisegliatin; Zabopegdutide; 64Cu-DOTA-AE105; TQA-3038; Amantadine Hydrochloride(SHINKEI Therapeutics); Mitoquinone mesylate; GAL-101; HS-10384; Vortosiran; Mitoxantrone hydrochloride liposome(Institute Of Hematology & Blood Diseases Hospital); Lipoic acid/Mecobalamin/Vitamin B1/Vitamin B6; WSD-0922; Deuterated vortioxetine; Emetine Hydrochloride; ETX-19477; HGP2102-1; HGP2102-2; Isocyclosporin A; Deuterated dimethyltryptamine; HGP-2102; GIM-531; CTO-0303; P4M-01; ITM-14D; Pozdeutinurad; Psilocybin(Pilz Bioscience); Dapagliflozin/Rosuvastatin (Cmg Pharmaceutical); R-Ketamine Hydrochloride Injection(Jiangsu Nhwa); DA-4505; Sustained released intravitreal implants(University of Kentucky); HY-072808; nL-CHCHD-001; AD-224; Montelukast oral film (IntelGenx); Calderasib; Iron sucrose (Renibus Therapeutics); 2000; Apomorphine(Grupo Ferrer Internacional); RS-5614; Ricorfotide vedotin; Tobramycin/Edetate Calcium sodium; [18F]AlF-NOTA-PCP2; Baxdrostat/dapagliflozin (AstraZeneca); NJ-2021-002; NRT-023; DW-5121; OATD-01; TQA-3810; NBI-1070770; Acetylcysteine lysinate; GNS-212-E; DWJ-1609; Ganaplacide/Lumefantrine; HSK-39775; Nature-derived psilocybin(Psyence Biomedical); NN-9505; Chylobinoid(Synthonics); AUR-109; ATX-01 (Arthex Biotech); BW-00112; Mesocaine; Psilocybin(Incannex); IMM-6-415; Colchicine/Ropivacaine; AD-223; RX-0301; AT-1965; FMC-376; VR-AD-1005; Mitucapistat; VH-4524184; DWC-202301; Nafamostat intravenous (Lowell Therapeutics); IVMED-85; MBF-015; KJ-14002; Mitoxantrone hydrochloride liposome (Zhongnan Hospital); Orziloben; FM-888; Lidocaine (Orexa); WXSH-0150; TY-0540; AB-001 (Agastiya Biotech); 177Lu-HTK03170; 68Ga-HTK03149; LDN-051; Aldifen; VI-0809; VI-0609; VI-0810; Bendamustine (Exinda); ATB-101; Al18F-NOTA-Pentixafor; Vezocolmitide; Meloxicam (Viatris); Toviblideg; GNP; CTO-1681; SIPI-6398; Zeptenstat; HP-518; Voclosporin (Qilu Pharmaceutical); [177Lu]JH020002; HYP-2090-PTSA; FB-849; BRS201; IMP-1734; OP-2024-C; CHF-6333; Cabamiquine; Avenanthramides; Varenicline Oxalate; CC-42344; TRM-270; Branch Chain Amino Acid(Mahidol University); Kamuvudines; AD-04(ADvantage Therapeutics); CRD-4730; AT-004(Arctic Therapeutics); AT-003(Arctic Therapeutics); Cyproheptadine Hydrochloride/Prazosin Hydrochloride; AL-8326; AL01211; VH-4004280; Fremocapavir; GSK-4524101; BGB-15025; 99mTc-CXCR4; F-18 Florastamin; Oral Arsenic Trioxide (Rasayani Biologics); BN-104; dapagliflozin formate; Rosuvastatin liposome encapsulated therapy (Beijing Inno Medicine); Atropine; Lysine-3,4-Methylenedioxymethamphetamine; Lenalidomide subcutaneous infusion (Starton Therapeutics); RGRN-305; DM-5167; HRF-2105; Lumacaftor (Qanatpharma); HLK-1004; HLK-1001; ATX-304; Vedroprevir; AZD9550; Brexanolone (extended-release injectable aqueous suspension formulation); TR-012001; Inlexisertib; Psilocybin(Apex Laboratories); K-833; K-757; Bilastine/Dextromethorphan Hydrobromide/Phenylephrine Hydrochloride; Cridanimod; Vanoglipel; Admilparant; Tuvusertib; FWD-1802; BBT-207; BB-1511; Tasipimidine; QLM-3004 (Qilu Pharmaceutical); Relugolix Combination; Sirolimus inhaled (OrphAI Therapeutics); Montelukast Gel(Aitiya (Shanghai) Pharma); Orellanine; Pyragrel Sodium; 177Lu-DOTA-EB-TATE; Relutrigine; Surlorian; Tuvutromstat; Ontunisertib; Ferric Pyrophosphate Liposomal; Ferrous ascorbate; EM-113; JIN-A02; Sutezolid; HRS-9950; TSN-222; Thymosin alpha 1; ILB-2109; HTL-0039732; D3S-002; TAK-733; PB-718; Octreotide; GTAEXS-617; ENX-102; BW-20507; IN-C036; NST-1024; NVP-2203; JZP-541; R2R01; ART6043; Mirivadelgat; Nacresertib; NS-050/NCNP-03; XY-0206; NGI-226; TNG-260; KNP2002; Zirdafulven; RMP-A-03; Vilzemetkib; Photodynamic therapy (Molteni Therapeutics); TQB-3728; RHH646; BRM-424; BBP-418; ENERGI-F703; PGN-EDO51; QY-101; CGT-1881; AZD-2693; Sarconeos; Tranexamic Acid (Bio54); Albuterol sulfate/fluticasone propionate (Teva Branded Pharmaceutical Industries); Prifemilast; Butaselen; BR-1733; 50561; CPL-01; TFX-06; HWH-340; ARINA-1; Pruvonertinib; XH-5102; Sodium Hyaluronate(Shinpoong); MH-080; ART-501; Enitociclib; DH-001; GEn1E-1124; RMG-03; Narazaciclib; INX-315; Pumecitinib; C-188-9; Phenylephrine hydrochloride (Talphera); ABBV-668; Nemtabrutinib; HST-1011; ADVC-001; Namodenoson; Levamlodipine Besylate/Valsartan (Sunshine Novo); SNP-ACTH (1-39) Gel; Ropivacaine extended release (PainReform); Panosyl-isomaltooligosaccharide; Clifutinib Besylate; Ciclosporin Eye Drops(CZhuhai Essex Bio-Pharma); Tianeptine Oxalate; donepezil (Vyant Bio); DWC202206; DWC202207; SC-0191; Atidafonat tosylate; Puliginurad; 18F-OP-801; Itruvone; Stimulan-VG; 99mTc-NDX-3315; Alpha-methyl-4-deoxy-4-[(18)F]fluoro-D-glucopyranoside; THDBH130; CBP-1019; Theophylline (Cyrano Therapeutics); Delocamten; Vabametkib; Adrixetinib; OM002; Yttrium-90 Carbon Microspheres; Serdexmethylphenidate; ALN-PNP; Galeflaprit; Ursodeoxycholic acid (Santen Pharmaceutical); Avenanthramide(Ceapro); CU-06; Iadademstat; JAB-2485; Suvadronabinol; CKD-498; Budesonide Sustained-release Capsules(Everest Medicine); GN-037; Alpibectir; DLQ-01; HY-3000; Icerguastat; LPM-3480392; LNK-01003; CKD-331; SYL-1801; Glasmacinal; Dabogratinib; GH-35; Zevotrelvir; KIO-301; Tofacitinib citrate (CAGE Bio); cRGD-ZW800-1; ABD-3001; Tebapivat; Ibogaine; Funobactam; Psilocybin infusion (Beckley Psytech); Empagliflozin/Sitagliptin Hydrochloride; DN-1508052; RP-1000; Linustedastat; Tigulixostat; Camlipixant; Nitrosooxypropanol; [11C]CPPC; HEC-169096; ESMESOL; Cambritaxestat; TT-301; EP-547; 68Ga-pentixafor; AGX-201; UI026; ASC-41; NRC-2694; [ 161 Tb]Tb PSMA I&T; EVO-101; Ceralasertib; Bofutrelvir; ML-004; R-906289 Monosodium; BR-790; ABI-2280; HCP-2102; Zeta-BC-003; D-4517; Singletine; Trichloroacetic acid; QBS-10072-S; OPL-0401; Diazo-oxo-L-norleucine; Neumifil(Pneumagen); Paclitaxel trevatide; RPN-301; 64Cu-SAR-BBN(Clarity Pharmaceuticals); MG-O-1002; Atorvastatin/Fenofibrate; VVN-539; RNK-05047; CDR-132L; D-xylitol/D-glucose/L-carnitine; Decitabine/Tetrahydrouridine (EpiDestiny/Novo Nordisk); GW-117; Kinezodianone R hydrochloride; DYP-688; K-161; Tranexamic acid (Leading BioSciences); TERN-501; Levonorgestrel/Meloxicam (InnovaGyn); Celecoxib/Ciprofloxacin; Palacaparib; QRX-003; kavalactones; BEBT-209; Tinodasertib; Bupivacaine implant; TFX-05-01; Cyclosporine/Loteprednol Etabonate; Zanvipixant; Irbesartan/Propagermanium; EN-002; MK-1088; Elzovantinib; ZG-19018; NMX-1; ACD-440; Quetiapine (Qrono); Histamine glutarimide; Velufenacin; SB-01 (Ensol BioSciences); Bocodepsin; CT-102; PTM-001 (Phoenicis Therapeutics); Valproic acid (Cereno Scientific); Lithium cocrystal; T3P-Y058-739; Halobetasol/lidocaine (Citius Pharmaceuticals); Sanfetrinem cilexetil; DNL-151; Vilagletistat; JBI-802; Nesuparib; Inaxaplin; RGT-075; Zatolmilast; TAS-119; ERAS-601; Atropine Sulfate Eye Drops(Zhaoke (Guangzhou) Ophthalmology Pharma); Atamparib; Methyl-beta-Cyclodextrin; Methylprednisolone sodium succinate (Nihon Pharmaceutical); Psilocybin; HS-10375; H-002; JX11502MA; ADPT-06; FG-001; Levothyroxine Sodium/Liothyronine sodium; Frondanol; Fulimetibant; BH-011; 68Ga-HA-DOTATATE; Lutetium-177 zadavotide guraxetan; Telmisartan/Verapamil Hydrochloride; Nanosilver Fluoride; RAD-105; RAD-102; RAD-104; ARO-C3; Anvumetostat; Isomyosamine; A-197; CNP-104; Brilaroxazine; CPL207-280CA; Florzolotau; ST-1703; Codivir; Deoxycholic Acid (Noratech Pharmaceuticals); Danifexor; Sacibertinib; PZH-2111; 1.0% povidone-iodine ophthalmic gel sterile solution (IVIEW Therapeutics); EG-017; RBD-4988; MN-08; Carbon monoxide; Irpagratinib; Pyrilutamide; TRV-734; MT-921; HR-19042; XTR-003; Fluoropezil; Obicetrapib; Piperine; Mitizodone Phosphate; CCX-587; PXS-6302; Agomelatine (Alto Neuroscience); MH-048; Zectivimod; ION-736; Palmitoylethanolamide; DWKH; Zinc oxide/Bismuth subgallate/Balsam peru/Bismuth oxide; Levodopa/Carbidopa controlled release tablets(WD Pharmaceutical); EF-175; AD-207; AD-202; Sumifilam; NBT-NM108; [18F]RP-115; BT-7480; Domiphen bromide/miconazole; Guanabenz Acetate; HA121-28; Soticlestat; ST-01; Elpipodect; Imdatifan; Prospekta; LY-356318; CS-02; KI 1115; KI 3108; KI 1114; PB-201; SEP-4199; HS-10376; Nitroxoline (Asieris Pharmaceuticals); HYML-122; PA-1010; Ceperognastat; Buloxibutid; Nefextinib hemifumarate; Reboxetine (Axsome Therapeutics); PCN-101; Mazindol Extended Release (NLS); Selonabant; Palmitoylethanolamide/Polydatin; ATX-101 (APIM Therapeutics); EQU-001; Evenamide Hydrochloride; Zifaxaban; SXR-1096; Merigolix; Lanifibranor; Taisi; Tamuzimod; EV-077; BMS-986166; Selatogrel; Ketotifen/Indomethacin; Romaciclib; Atuzabrutinib; AB-2004; Ga-68 Dolacga; AD-113; 177Lu-FAP-2286; Angiontensin(1-7); TRV-120027; NNC-0165-1875; AP-L1898; 18F vipivotide tetraxetan; MRX-2843; Olanzapine transdermal patch (Starton Therapeutics); YG-1699; Tipiracil Hydrochloride; Ulefnersen; KH-001; Manukapli(Manukamed); DX1002; Perindoprilat; Paracetamol; 99m-TC-PSMA-I&S; SHR0410; Dexlipoic acid lysine; 18-Methoxycoronaridine; Bemnifosbuvir; Dapagliflozin formate/Linagliptin; Avenciguat; Inidascamine; SP5M-001; SJ-557733; FCN-011; Lu-177-DGUL; Ga-68-NGUL; NFL-101; Sodium Pyruvate; Emilumenib succinate; Atropine sulphate (Ocumension Therapeutics); Ibogaine HCl (ATAI Life Sciences/DemeRx); QLS-101; Alogabat; Runcaciguat; DBI-002; LU-177-SSTR- PNT-2003; Tideglusib; 64Cu-SarTate; PF-06412562; tamsulosin; Liposomal Cetirizine; Selvigaltin; Dapagliflozin/Pioglitazone; S-fluoxetine; R-fluoxetine; Dimolegin; Larotinib Mesylate; Gallium-68-DOTA-minigastrin; Edralbrutinib; Belvarafenib; DSP-2230; AS-012; Chloroquine Phosphate Gel(Hybribio Biotech); RDX-013; Mycophenolic Acid/Betamethasone Sodium Phosphate; Ecdysterone; Exenatide oral (Oramed); Germinal Peptide; HOV-12020; Amsulostat; Idrebormilast; Vepafestinib; Axitinib injectable suspension (Clearside Biomedical); kisspeptin 112-121; MT-1002(Shaanxi Micot Technology); APSCTC; Diclofenac sodium transdermal patch (Hisamitsu Pharmaceuticals); Nicotinamide riboside/Pterostilbene; Resiniferatoxin; AGN-193408; MC-0518; CX13-608; DAW-2020; Zagociguat; BHV-1100; Pizuglanstat; Traneurocin; CNM-ZnAg; LY-3130481; A9T-1101; rineterkib; Rezatapopt; Hypochlorous Acid; ApTOLL; Timolol maleate gel (Auson Pharmaceuticals); AZD-8233; HCP-1904; BEN-2293; Lidocaine/Heparin; Metablok; SX-682; Udonitrectag; Rutan; Dexfenfluramine Hydrochloride; SHR-2150; Fesomersen; Pilavapadin; NT-219; Articaine ophthalmic (American Genomics); 2-FL; AK-1830; Isuzinaxib hydrochloride; ACC-006; NFX-179; MM-II; ocifisertib; Tianagliflozin; NX-9; Petadeferitrin; Dalzanemdor; THR-149; Efocipegtrutide; CNM-Au8; ARO-ENaC; Ifenprodil (Algernon Pharmaceuticals); Metyrapone/Oxazepam; CVI-LM-001; Pulrodemstat; AZR-MD-001; Oremepermin alfa; Miconazole (Hill Dermaceuticals); EA4000; Firibastat; BAY-85-8102; Vidofludimus calcium; Etrinabdione; Vamifeport hydrochloride; XNW-7201; Etrumadenant; Radspherin; HTMC-0435; Temuterkib mesylate; IFM-2427; BGB-10188; SHC014748M; Acarbose/Orlistat; EF-009; Amitriptyline oxalate; ST-617; N-acetylglucosamine; Sinapultide; Dasminapant; Amlodipine/Telmisartan/Indapamide; SVT-15652; SRP-100; Bafrekalant; ASC09F; AUR-101; Linezolid intradiscal (Persica Pharmaceuticals); TBA-7371; Miramistin; BRM-421; Azacitidine (Boryung Pharmaceutical); Nuvisertib; Fisogatinib; Minerval; Sucunamostat; Dexamethasone sodium phosphate sustained release (Taiwan Liposomal Company); Nuzefatide pevedotin; Venadaparib; Zotatifin; Idroxioleic acid; Alprostadil Liposome for Injection(CSPC Zhongqi Pharma); Siremadlin; JNJ-54175446; Deudomperidone; AP-30663; CLE-100; Praziquantel paediatric formulation (Pediatric Praziquantel Consortium); CTB-02; OLX-10010; Taniborbactam; Hemay007; QL-007; Rogaratinib; Cimdelirsen; Lenumlostat hydrochloride; Aminoarteether Maleate; Lutetium (177Lu) zaregreptide dizuxetan; Vociprotafib; Fosdesdenosine sipalabenamide; Lopinavir/Ritonavir/Lamivudine/Zidovudine; Zamicastat; TK-112690; Teriflunomide Sodium; Lutetium-177 DOTA satoreotide; Gildeuretinol; Rifaquizinone; D-0120-NA; Serlopitant; ODM-209; Foxy-5; VK-2019; Sepofarsen; Gacyclidine; Nutraquinol; Norketotifen; Pramipexole/Aprepitant; Ganfeborole; Nedisertib; Cevidoplenib; OMT-28; Gamma-Tocotrienol; Diflucortolone Valerate Cream(Tianjin Pharmaceutical Research Institute); JBPOS-0101; Bavdegalutamide; Matsupexole; Fasudil (Raya Therapeutic); Patidegib; Ridinilazole; Ampreloxetine; Tominersen; ODN/Pam2; NRP-2945; BR-2251; Ruxotemitide; Nitazoxanide (Genfit); Ralmitaront; Abivertinib; Zifogaptide; Carbetocin intranasal (Ferring Pharmaceuticals); JAB-3068; 11C-UCB-J; Opelconazole; LTM-1201L; Lixosicone; Fosifloxuridine nafalbenamide; Diclofenac sodium gel (Amzell); Subasumstat; Pramipexole/Ondansetron; LYS006; [11C]ER-176; Fostroxacitabine bralpamide; DLBS-2411; Bevantolol-hydrochloride (SOM Biotech); 18F-BMS-986229; Foslinanib; Lucerastat; [18F]PSMA-11; Zelquistinel; Cannabidiol Gel (Zynerba); Selumetinib sulfate/MK-2206; Capsaicin (Propella Therapeutics); BEY-1107P; Dexamethasone/Netilmicin Sulfate; Huperizine-A (Biscayne Pharmaceuticals); Selgantolimod; GLWL-01; Zetomipzomib; LH-8; DEP-Cabazitaxel; Tovinontrine; Seal oil omega-3 polyunsaturated fatty acid; Imarikiren hydrochloride; APT-5031; Compound aluminum sulfate; DAW1033D; Dexamethasone sodium phosphate injectable gel (Scilex Holding); Leriglitazone; Limantrafin; 68Ga-NODAGA-E[c(RGDyK)]2; Onvansertib; Samuraciclib; Envogmilast; Teroo Hydrochloride; Atuliflapon; Mosedipimod; (S,S)-[11C]MeNER; Apinocaltamide; Vorbipiprant sodium; Tramadol (Avenue Therapeutics); SJP-0125; CN-105; H3B-6545; Clesacostat; TS-121; Nangibotide; Lacripep; Vilaprisan; Indisetron Dihydrochloride; Ipatasertib; PXS-4728; KRP-116D (Kyorin Pharmaceutical); Tivanisiran; Netupitant; PT-2385; Ibuprofenamine Hydrochloride; Dapolsertib hydrochloride; [18F]F-AraG; Hematoporphyrin Ether Ester; LM11A-31; Cotsiranib; Delpazolid; Amelparib; Ibrilatazar; Mesdopetam; PDMX-1001; Pesampator; M-7583; TOL-463; Fimepinostat; Soclenicant; Genipin; Vodobatinib; DUK-CPG-001; Pravibismane; Merestinib; Prexigebersen; ivaltinostat; Phospholipovit; HTB-003; Idasanutlin; Plinabulin; Tilsotolimod; Apabetalone; Azilsartan Trimethylethanolamine; GSK-2256098; Abimufloxacin; Pirotinib Hydrochloride; YH-12852; Berzosertib; Atorvastatin Calcium Hydrate/Levamlodipine; BAY-94-9392; Rhenium (186Re) obisbemeda; Taselisib; Danvatirsen; Ethylmethylhydroxypyridine Succinate; Cannabidivarin; Varoglutamstat; Atorvastatin Calcium Hydrate/Hyzetimibe; Prexasertib; Isoquercetin; Bifonazole/Triamcinolone Acetonide; CC-10015; Potassium-Hydroxypentyl Benzoate; Leuprorelin depot(Camurus); Dexamethasone intravitreal implant (Aerie Pharmaceuticals); DHL-HisZnNa(Oita University); Imifoplatin; Cinhyaluronate sodium; Mirabegron/Solifenacin Succinate; Imidol Hydrochloride; Vincristine Sulfate Liposome; Tyroservaltide; Tetrodotoxin; Basmisanil; Tilidine Hydrochloride/Naloxone; Veliparib Hydrochloride; Lidocaine/Allantoin/Glycyrrhetinic Acid/Vitamin E; Ciraparantag; Galunisertib; Implantable sustained-release cisplatin (Zhongren Technology); Oltipraz; 5-aminolevulinic acid hydrochloride/Sodium ferrous citrate; Ambroxol Hydrochloride/Salbutamol sulfate; Ceftazidime/Sulbactam sodium; Methylprednisolone aceponate (Tianjin Pharmaceutical Research Institute); Cebranopadol hemicitrate; 188Re-HEDP; Tocopheryl phosphate mix (Phosphagenics); Oxytocin (Tonix Pharmaceuticals); Allantoin; Rimiducid; Ulixertinib; 129Xe; Picropodophyllin; Metacavir; Galeterone; LY-2940094; Buparlisib; Icenticaftor; Solnatide; IPP-204106; Foscenvivint; Gandotinib; Itacitinib; Olaptesed Pegol; [11C]PBR-28; Osteodex; Cipargamin; Modified Sodium Montmorillonite; Triciribine Phosphate; Antineoplaston As2-1/Antineoplaston A10; Quisinostat Hydrochloride; Apitolisib; Dactolisib; Ifetroban; Methoxyflurane; Epetraborole; ADX-71149; Biperiden Hydrochloride; Ferric Pyrophosphate Citrate; Dexpramipexole Dihydrochloride; Censavudine; Crolibulin; Guadecitabine Sodium; Eptazocine hydrobromide; Pentazocine; CBL-0137; Mometasone eluting resorbable scaffold (Lyra Therapeutics); L-Demethyl Phencynonate Hydrochloride; Onvapegleukin alfa; CF Combo; Staccato Alprazolam(Engage ); Basimglurant Sulfate; Nitroglycerin(Damascus University); UI028; Yogliptin; MTL-CEBPA; 225Actinium-PSMA-I&T; SYHA1402; YPS-345; Tosposertib phosphate; Verenafusp alfa; LPCN-1148; Tramadol Hydrochloride/Etoricoxib; NNC0480-0389; Oral Denatonium Acetate(Aardvark); Chlorine dioxide (Tarsus Pharmaceuticals); JW-0101; C-2101; LivaloVA; KL-130008; Levofloxacin/Ketorolac Tromethamine; NMBS-2; PIN-201104; IMP-9064; SM-020; Dexamethasone ophthalmic (Oculis Pharma); Ketoprofen/Gabapentin; Oral Edaravone (Treeway); RP-7214; Dazdotuftide; NLM-001; Sodium tungstate (Oxolife); Hydroxychloroquine sulfate/Sirolimus; Epivotide; MHV-370; Onfasprodil; Bilastine/Montelukast; Asengeprast; 18F-92; Ecubectedin; Mefuparib Hydrochloride; Celecoxib/Famciclovir; Epaldeudomide; SNB-011; Adiponectin analogue (Allysta Pharmaceuticals); CPL-500036; Valiltramiprosate; MIB-626; CBX-12; Medical Cannabis(Syqe Medical); Timolol ophthalmic (Betaliq); Nebivolol ophthalmic (Betaliq); Amdizalisib; GL-101; Eclitasertib; Govorestat; Chiauranib; Antarelix; Salfaprodil; BI-474121; Mobinitinib fumerate; PIPE-505; Fosgonimeton; NKP-1339; Firzacorvir; AMXI-5001; Cronexitide lanocianine; Redasemtide; AZD-6482; CG001419; Clonidine; GRWD-5769; Olisutrigine bromide; DC-806; SPH-4336; Naltrexone Implants (Shenzhen Sciencare Medical Industries ); BBT-877; AMZ-002; ICP-490; LY-5625574; TP-1222; SC-0245; AC01; Divesiran; [68-Ga]CBP-8; JW-0201; Paclitaxel/Hyaluronic acid; Azilsartan mepixetil Potassium; KI-0503; Deucrictibant; Napazimone; Cenerimod; Clobetasol propionate ophthalmic nanoemulsion (Salvat); TPM-502; Salvianolic acid A (Shanghai Pharmaceuticals Holding); AMXT-1501; Sulforafan alfadex; AZD-5069; Voxvoganan; MK-2206; Resveratrol; Resiquimod; Leflutrozole; Doxorubicin in P-glycoprotein-targeting pluronics(Christie Hospital Nhs Foundation Trust); Milciclib maleate; Burixafor Hydrobromide; BNC-105P; Linsitinib; Phosphatidyl choline; VB-201; Pimasertib hydrochloride; Vilanterol Trifenatate; Tetrahydrouridine; FdCyd; Cu(II)ATSM; Firtecan pegol; Telatinib; Sapitinib; AUS-131; Pradigastat; Alisertib; Rigosertib Sodium; AZD-1656; Alvelestat; CBP-501; Fluridil; Anacetrapib; CD-4802; Efatutazone hydrochloride; Nabilone; Tasquinimod; Muparfostat sodium; E-7820; Nadolol; 2-Deoxyglucose

Data notes

  • Sales column: ▲ = observed global peak sales, * = public estimate, blank = no sales data. Cross-verified against public revenue figures, so the unit is USD billion.
  • Expiry years are public compound/core patent expiries (US); patent-library-level per-year verification happens at onboarding.
  • Semaglutide (peptide biologic) is outside the chemical-drug search scope, so it is not listed here; its sidechain intermediates are covered separately in the LOE opportunity library.
  • Dapagliflozin / canagliflozin matched metformin combination products, not the single agent.
  • Biologics have no synthetic intermediate chain, so the impact on intermediate mapping is limited.

Source: cross-verified sources · window 2028-2033 · generated 2026-10-22 · Sales unit: USD billion (cross-verified)