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Cabamiquine

Tier C — Watch / trade

Cabamiquine

University Of Dundee
Originator
-
First approval
-
Expiry (public)
No sales data
Peak sales
Small molecule
Type

Targets:EF2

Indications (approved):Plasmodium infection

Regional status

US
-
EU
No progress
2020-02-17
China
-
Japan
-

Synthetic routes & intermediates2 routes

Originator routes × 1Optimised (non-patent) × 1Process routes × 0

Routes are ordered originator first, then optimised / process (non-patent) routes; each lists steps, overall yield and the intermediate table (code / CAS / name) — ready for supplier sourcing and RFQ. Rendered by this site from structured data; no third-party route graphics used.

OriginatorRoute 1Steps 4 · Total yield 625 mg
M-5717-00117201-43-3M-5717-00237812-51-4M-5717-003265107-94-6M-5717-004443-69-6M-5717-0051469440-03-6M-5717-0067154-73-6API · Cabamiquine
CodeCAS No.Intermediate
M-5717-00117201-43-34-(bromomethyl)benzonitrile
M-5717-00237812-51-44-(morpholinomethyl)benzonitrile
M-5717-003265107-94-61-(4-(morpholinomethyl)phenyl)ethan-1-one
M-5717-004443-69-65-fluoroindoline-2,3-dione
M-5717-0051469440-03-66-fluoro-2-(4-(morpholinomethyl)phenyl)quinoline-4-carboxylic acid
M-5717-0067154-73-62-(pyrrolidin-1-yl)ethan-1-amine
OptimisedRoute 2Steps 6 · Total yield 0.6 g
M-5717-007607-40-9M-5717-0081885123-22-7M-5717-0091469439-99-3M-5717-010364794-79-6M-5717-011589-15-1M-5717-012132833-51-3API · Cabamiquine
CodeCAS No.Intermediate
M-5717-007607-40-96-fluoro-2-hydroxyquinoline-4-carboxylic acid
M-5717-0081885123-22-72-chloro-6-fluoroquinoline-4-carbonyl chloride
M-5717-0091469439-99-32-chloro-6-fluoro-N-(2-(pyrrolidin-1-yl)ethyl)quinoline-4-carboxamide
M-5717-010364794-79-6Available4-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzyl)morpholine
M-5717-011589-15-11-bromo-4-(bromomethyl)benzene
M-5717-012132833-51-34-(4-bromobenzyl)morpholine

Frequently asked questions

What are the approved indications of Cabamiquine?

Approved indications include: Plasmodium infection.

When does the Cabamiquine patent expire?

No public expiry year is available for Cabamiquine yet; this page updates once verified.

How many synthesis routes are recorded for Cabamiquine?

2 synthesis routes are recorded; the shortest is 4 steps with 625 mg total yield. Intermediates in each route carry codes and CAS numbers.

Where can I buy Cabamiquine intermediates?

1 intermediate CAS of Cabamiquine are available through the Unibest supply network — see the route tables on this page and request a quote per CAS.

How do I get a quote for Cabamiquine intermediates?

Open the CAS profile of the target intermediate from this page, or submit an RFQ directly — the CAS enters the matching flow automatically and the supply network responds with quotes.

Source: cross-verified data (structured fields only) · 2026-10-22