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Tianagliflozin

Tier C — Watch / trade

Tianagliflozin

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Originator
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First approval
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Expiry (public)
No sales data
Peak sales
Small molecule
Type

Targets:SGLT2

Indications (approved):Type 2 diabetes

Regional status

US
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EU
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China
Phase II
2020-08-10
Japan
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Synthetic routes & intermediates1 routes

Originator routes × 1Optimised (non-patent) × 0Process routes × 0

Routes are ordered originator first, then optimised / process (non-patent) routes; each lists steps, overall yield and the intermediate table (code / CAS / name) — ready for supplier sourcing and RFQ. Rendered by this site from structured data; no third-party route graphics used.

OriginatorRoute 1Steps 6 · Total yield /
Tianagliflozin-001461432-26-8Tianagliflozin-0021590387-75-9Tianagliflozin-0031415905-90-6Tianagliflozin-0041443341-94-3Tianagliflozin-0051590387-76-0Tianagliflozin-0061590387-77-1API · Tianagliflozin
CodeCAS No.Intermediate
Tianagliflozin-001461432-26-8(3R,4R,5S,6R)-2-(4-chloro-3-(4-ethoxybenzyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol
Tianagliflozin-0021590387-75-9(2R,3S,4R,5R,6S)-2-(((tert-butyldimethylsilyl)oxy)methyl)-6-(4-chloro-3-(4-ethoxybenzyl)phenyl)tetrahydro-2H-pyran-3,4,5-triol
Tianagliflozin-0031415905-90-6(2R,3R,4R,5S,6S)-2-(((tert-butyldimethylsilyl)oxy)methyl)-6-(4-chloro-3-(4-ethoxybenzyl)phenyl)tetrahydro-2H-pyran-3,4,5-triyl triacetate
Tianagliflozin-0041443341-94-3(2S,3S,4R,5R,6R)-2-(4-chloro-3-(4-ethoxybenzyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triyl triacetate
Tianagliflozin-0051590387-76-0(2S,3S,4R,5S,6S)-2-(4-chloro-3-(4-ethoxybenzyl)phenyl)-6-(iodomethyl)tetrahydro-2H-pyran-3,4,5-triyl triacetate
Tianagliflozin-0061590387-77-1(2S,3S,4S,5R,6R)-2-(4-chloro-3-(4-ethoxybenzyl)phenyl)-6-methyltetrahydro-2H-pyran-3,4,5-triyl triacetate

Frequently asked questions

What are the approved indications of Tianagliflozin?

Approved indications include: Type 2 diabetes.

When does the Tianagliflozin patent expire?

No public expiry year is available for Tianagliflozin yet; this page updates once verified.

How many synthesis routes are recorded for Tianagliflozin?

1 synthesis routes are recorded; the shortest is 6 steps with / total yield. Intermediates in each route carry codes and CAS numbers.

Where can I buy Tianagliflozin intermediates?

All intermediates in Tianagliflozin routes have CAS profiles — you can submit an RFQ per CAS and it enters the Unibest matching pool.

How do I get a quote for Tianagliflozin intermediates?

Open the CAS profile of the target intermediate from this page, or submit an RFQ directly — the CAS enters the matching flow automatically and the supply network responds with quotes.

Source: cross-verified data (structured fields only) · 2026-10-22