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Ifupinostat Hydrochloride

Tier C — Watch / trade

Ifupinostat Hydrochloride

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Originator
2025
First approval
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Expiry (public)
No sales data
Peak sales
Small molecule
Type

Targets:Class I PI3K, HDAC

Indications (approved):Diffuse large B-cell lymphoma

Regional status

US
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EU
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China
Approved
2025-06-30
Japan
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Synthetic routes & intermediates1 routes

Originator routes × 1Optimised (non-patent) × 0Process routes × 0

Routes are ordered originator first, then optimised / process (non-patent) routes; each lists steps, overall yield and the intermediate table (code / CAS / name) — ready for supplier sourcing and RFQ. Rendered by this site from structured data; no third-party route graphics used.

OriginatorRoute 1Steps 12 · Total yield 10.04 kg (BEBT-908)
BEBT-9081646906-27-5BEBT-908-00122288-78-4BEBT-908-00216233-51-5BEBT-908-00316234-14-3BEBT-908-00416234-15-4BEBT-908-005885618-31-5BEBT-908-006955979-15-4BEBT-908-00789793-12-4BEBT-908-0081235450-25-5BEBT-908-009265664-53-7BEBT-908-0101339926-04-3BEBT-908-0111235449-52-1BEBT-908-012624-28-2BEBT-908-01384539-30-0BEBT-908-014227939-01-7API · Ifupinostat Hydrochloride
CodeCAS No.Intermediate
BEBT-9081646906-27-5N-hydroxy-2-(methyl((2-(6-(methylamino)pyridin-3-yl)-4-morpholinothieno[3,2-d]pyrimidin-6-yl)methyl)amino)pyrimidine-5-carboxamide trihydrochloride
BEBT-908-00122288-78-4methyl 3-aminothiophene-2-carboxylate
BEBT-908-00216233-51-5thieno[3,2-d]pyrimidine-2,4(1H,3H)-dione
BEBT-908-00316234-14-32,4-dichlorothieno[3,2-d]pyrimidine
BEBT-908-00416234-15-44-(2-chlorothieno[3,2-d]pyrimidin-4-yl)morpholine
BEBT-908-005885618-31-52-chloro-4-morpholinothieno[3,2-d]pyrimidine-6-carbaldehyde
BEBT-908-006955979-15-41-(2-chloro-4-morpholinothieno[3,2-d]pyrimidin-6-yl)-N-methylmethanamine
BEBT-908-00789793-12-4Availableethyl 2-chloropyrimidine-5-carboxylate
BEBT-908-0081235450-25-5ethyl 2-(((2-chloro-4-morpholinothieno[3,2-d]pyrimidin-6-yl)methyl)(methyl)amino)pyrimidine-5-carboxylate
BEBT-908-009265664-53-7(6-(methylamino)pyridin-3-yl)boronic acid hydrochloride
BEBT-908-0101339926-04-3ethyl 2-(methyl((2-(6-(methylamino)pyridin-3-yl)-4-morpholinothieno[3,2-d]pyrimidin-6-yl)methyl)amino)pyrimidine-5-carboxylate
BEBT-908-0111235449-52-1N-hydroxy-2-(methyl((2-(6-(methylamino)pyridin-3-yl)-4-morpholinothieno[3,2-d]pyrimidin-6-yl)methyl)amino)pyrimidine-5-carboxamide
BEBT-908-012624-28-22,5-dibromopyridine
BEBT-908-01384539-30-05-bromo-N-methylpyridin-2-amine
BEBT-908-014227939-01-7tert-butyl (5-bromopyridin-2-yl)(methyl)carbamate

Frequently asked questions

What are the approved indications of Ifupinostat Hydrochloride?

Approved indications include: Diffuse large B-cell lymphoma.

When does the Ifupinostat Hydrochloride patent expire?

No public expiry year is available for Ifupinostat Hydrochloride yet; this page updates once verified.

How many synthesis routes are recorded for Ifupinostat Hydrochloride?

1 synthesis routes are recorded; the shortest is 12 steps with 10.04 kg (BEBT-908) total yield. Intermediates in each route carry codes and CAS numbers.

Where can I buy Ifupinostat Hydrochloride intermediates?

1 intermediate CAS of Ifupinostat Hydrochloride are available through the Unibest supply network — see the route tables on this page and request a quote per CAS.

How do I get a quote for Ifupinostat Hydrochloride intermediates?

Open the CAS profile of the target intermediate from this page, or submit an RFQ directly — the CAS enters the matching flow automatically and the supply network responds with quotes.

Source: cross-verified data (structured fields only) · 2026-10-22