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CAS 506-59-2
Dimethylamine hydrochloride
登记编号：Carteolol Hydrochloride-015、Desvenlafaxine-035、(XII) 920279-2-a、(XI) 920279-3-a、(VIII) 920279-4-a、(II)145089-15-a
应用背景（按来源药适应症）
高眼压盐酸卡替洛尔/拉坦前列素青光眼盐酸卡替洛尔/拉坦前列素开角型青光眼盐酸卡替洛尔/拉坦前列素重度抑郁症地文拉法辛抑郁症地文拉法辛高血压盐酸卡替洛尔高眼压盐酸卡替洛尔青光眼盐酸卡替洛尔心绞痛盐酸卡替洛尔心律失常盐酸卡替洛尔非小细胞肺癌甲磺酸兰泽替尼肝功能衰退甲磺酸兰泽替尼阿尔茨海默病重酒石酸卡巴拉汀痴呆重酒石酸卡巴拉汀帕金森病重酒石酸卡巴拉汀抗胆碱能综合征重酒石酸卡巴拉汀神经行为学表现重酒石酸卡巴拉汀认知障碍重酒石酸卡巴拉汀
来源药（使用该中间体的合成路线）
| 品种 | 梯队 | 到期年 |
|---|---|---|
| 盐酸卡替洛尔/拉坦前列素Carteolol Hydrochloride/Latanoprost | Tier C · 观察 / 贸易 | - |
| 地文拉法辛Desvenlafaxine | Tier C · 观察 / 贸易 | - |
| 盐酸卡替洛尔Carteolol Hydrochloride | Tier C · 观察 / 贸易 | - |
| 甲磺酸兰泽替尼Lazertinib Mesylate | Tier C · 观察 / 贸易 | - |
| 重酒石酸卡巴拉汀Rivastigmine Tartrate | Tier B · 提前布局 | - |
合成路线中的位置（上下游链）
按路线登记顺序排列，左→右为合成方向；高亮为当前 CAS，其余可点击跳转对应档案。
2-(Benzyloxycarbonylamino)acetic acid→Dimethylamine hydrochloride→Benzyl [2-(dimethylamino)-2-oxoethyl]carbamate→N,N-Dimethylglycinamide→Carboxyethane→N-[2-(Dimethylamino)-2-oxoethyl]propanamide→1-Iodo-2-methoxybenzene→N-[2-(Dimethylamino)-2-oxoethyl]-3-(2-methoxyphenyl)propanamide→2-(5-Methoxy-2-oxo-3,4-dihydroquinolin-1(2H)-yl)-N,N-dimethylacetamide
2-(4-Methoxyphenyl)acetonitrile→2-(4-Hydroxyphenyl)acetonitrile→[4-[(2-Methoxyethoxy)methoxy]phenyl]acetonitrile→Cyclohexanone→(1-Hydroxycyclohexyl)[4-[(2-methoxyethoxy)methoxy]phenyl]acetonitrile→Dimethylamine hydrochloride→Desvenlafaxine-036→4-[2-(Dimethylamino)-1-(1-hydroxycyclohexyl)ethyl]phenol→(1-Hydroxycyclohexyl)(4-hydroxyphenyl)acetonitrile
2-(Benzyloxycarbonylamino)acetic acid→Dimethylamine hydrochloride→Benzyl [2-(dimethylamino)-2-oxoethyl]carbamate→N,N-Dimethylglycinamide→Carboxyethane→N-[2-(Dimethylamino)-2-oxoethyl]propanamide→1-Iodo-2-methoxybenzene→N-[2-(Dimethylamino)-2-oxoethyl]-3-(2-methoxyphenyl)propanamide→2-(5-Methoxy-2-oxo-3,4-dihydroquinolin-1(2H)-yl)-N,N-dimethylacetamide
2-Amino-5-fluoro-4-nitroanisole→N-Boc-4-Fluoro-2-methoxy-5-nitroaniline→1-Oxa-4-azacyclohexane→N-Boc-2-Methoxy-4-morpholin-4-yl-5-nitroaniline→tert-Butyl [5-amino-2-methoxy-4-(morpholin-4-yl)phenyl]carbamate→(Chloromethyl)acetyl chloride→tert-Butyl [5-(3-chloropropanamido)-2-methoxy-4-(morpholin-4-yl)phenyl]carbamate→N-(5-N-Boc-Amino-4-methoxy-2-morpholin-4-ylphenyl)acrylamide→N-[5-Amino-4-methoxy-2-(morpholin-4-yl)phenyl]prop-2-enamide→1-(2-Chloropyrimidin-4-yl)-3-phenyl-1H-pyrazole-4-carbaldehyde→N-[5-[[4-(4-Formyl-3-phenyl-1H-pyrazol-1-yl)pyrimidin-2-yl]amino]-4-methoxy-2-(morpholin-4-yl)phenyl]prop-2-enamide→Dimethylamine hydrochloride→N-[5-[(4-[4-[(dimethylamino)methyl]-3-phenyl-1H-pyrazol-1-yl]pyrimidin-2-yl)amino]-4-methoxy-2-(morpholin-4-yl)phenyl]prop-2-enamide
2-Amino-5-fluoro-4-nitroanisole→1-Oxa-4-azacyclohexane→2-Methoxy-4-(morpholin-4-yl)-5-nitroaniline→2-Methoxy-4-morpholin-4-yl-5-nitrophenylformamide→5-Amino-2-methoxy-4-morpholin-4-ylphenylformamide→(Chloromethyl)acetyl chloride→3-Chloro-N-[5-formamido-4-methoxy-2-(morpholin-4-yl)phenyl]propanamide→N-[5-(Formylamino)-4-methoxy-2-morpholin-4-ylphenyl]acrylamide→1-[2-(Methanesulfonyl)pyrimidin-4-yl]-3-phenyl-1H-pyrazole-4-carbaldehyde→N-[5-[[4-(4-Formyl-3-phenyl-1H-pyrazol-1-yl)pyrimidin-2-yl]amino]-4-methoxy-2-(morpholin-4-yl)phenyl]prop-2-enamide→Dimethylamine hydrochloride→N-[5-[(4-[4-[(dimethylamino)methyl]-3-phenyl-1H-pyrazol-1-yl]pyrimidin-2-yl)amino]-4-methoxy-2-(morpholin-4-yl)phenyl]prop-2-enamide→3-Phenyl-1H-pyrazole-4-carbaldehyde→4-Chloro-2-(methylsulfanyl)pyrimidine→1-[2-(Methylsulfanyl)pyrimidin-4-yl]-3-phenyl-1H-pyrazole-4-carbaldehyde
本站可供应的对应中间体
同 CAS 多家在售供应横向对比；价格区间为供应方挂牌口径，实价以询价确认为准。
| 供应商 | 产品 | 价格区间 | 最小起订 | 货期 | 资质 | 操作 |
|---|---|---|---|---|---|---|
| Unibest Nantong cGMP Site | 3-phenyl-1H-pyrazole-4-carbaldehyde Pharmaceutical Intermediates | 询价 | 询价 | 询价 | — | |
| Unibest Taizhou GMP-like Site | 4-Chloro-2-(methylsulfonyl)pyrimidine Pharmaceutical Intermediates | 询价 | 询价 | 询价 | — | |
| Qualified Partner — East China API Works | 4-chloro-N-(2-methoxy-4-morpholino-5-nitrophenyl)pyrimidin-2-amine Pharmaceutical Intermediates | 询价 | 询价 | 询价 | — | |
| Unibest Nantong cGMP Site | 1-(2-((2-methoxy-4-morpholino-5-nitrophenyl)amino)pyrimidin-4-yl)-3-phenyl-1H-pyrazole-4-carbaldehyde Pharmaceutical Intermediates | 询价 | 询价 | 询价 | — | |
| Unibest Taizhou GMP-like Site | 4-(4-((dimethylamino)methyl)-3-phenyl-1H-pyrazol-1-yl)-N-(2-methoxy-4-morpholino-5-nitrophenyl)pyrimidin-2-amine Pharmaceutical Intermediates | 询价 | 询价 | 询价 | — | |
| Qualified Partner — East China API Works | N1-(4-(4-((dimethylamino)methyl)-3-phenyl-1H-pyrazol-1-yl)pyrimidin-2-yl)-6-methoxy-4-morpholinobenzene-1,3-diamine Pharmaceutical Intermediates | 询价 | 询价 | 询价 | — |
本页为中间体 CAS 注册档案：同 CAS 的多条路线登记已合并；后续供应商报价与买方需求以该 CAS 为主键撮合。